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2-[2-(1H-pyrazol-1-yl)ethyl]-4-(4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-cycloheptanecarbonylpiperidine
N-({6-[3-(morpholin-4-ylmethyl)phenyl]pyridin-3-yl}methyl)acetamide
(1S,5R)-6-(pyridin-2-ylmethyl)-3-{thieno[2,3-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-fluoroethyl)-5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazole
ethyl 1-(propylcarbamoyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-benzyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{[1-(ethanesulfonyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
5-(morpholin-4-ylmethyl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}furan-3-carboxamide
2-(3-fluorophenyl)-1-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
1-cyclopentanecarbonyl-N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]piperidine-4-carboxamide
8-{4-[(2-hydroxyethyl)(methyl)amino]piperidin-1-yl}-2,6-dimethyloctan-2-ol
ethyl 4-[4-(5-methyl-1,3-benzoxazol-2-yl)piperazin-1-yl]piperidine-1-carboxylate
1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
1-cyclohexanecarbonyl-4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-(2-methoxyethyl)-3,6-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1-benzofuran-2-carboxamide
(3R)-1-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}pyrrolidin-3-ol
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
7-fluoro-1-methyl-2-(4-propylpyrimidine-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline
2-cyclopropyl-9-[2-(4-fluorophenyl)-2-hydroxyacetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4-chlorophenyl)ethyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
3-{5-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-{4-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-4-(pyrrolidin-3-yl)benzamide
3-(pyridin-4-yl)-N-[2-(4-sulfamoylphenyl)ethyl]propanamide
6-(methoxymethyl)-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrimidin-4-amine
3-(3-methoxyphenoxymethyl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidine
6-(5-fluoro-2-methoxyphenyl)-2,4-dimethylpyridine-3-carbonitrile
1-[4-(furan-2-ylmethyl)piperazin-1-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
2-[2-(2-fluoro-4-methylphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
4-(4-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}-1H-1,2,3-triazol-1-yl)-N-propylpiperidine-1-carboxamide
N-benzyl-N-(4-hydroxybutyl)-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
5-butyl-1'-(pyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(2-chlorophenyl)methyl]-3-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}propanamide
4-[(dimethylamino)methyl]-1-(pyrimidin-4-yl)azepan-4-ol
N-{4-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}-4-[(methylsulfanyl)methyl]piperidine-1-carboxamide
2-[(5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-{4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}ethan-1-one
3-butyl-4-[3-(dimethylamino)benzoyl]-1-methylpiperazin-2-one
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine
4-(2-methyl-1H-imidazol-1-yl)-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidine-4-carboxylic acid
1,3-dimethyl-5-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}imidazolidine-2,4-dione
N-[2-(propan-2-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
3-({9-oxo-1-oxa-8-azaspiro[4.6]undecan-8-yl}methyl)benzonitrile
1-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-3-(furan-2-yl)propan-1-one
N-cyclopropyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
[(3R,4S)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
6-{4-[(3,5-dimethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-2-carbonitrile
6-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]pyridine-3-carbonitrile
2-methyl-6-{[3-(5-methylfuran-2-yl)butyl]amino}heptan-2-ol
2-[({5-[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol