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N,N-diethyl-1-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-3-carboxamide
(3R,4R)-1-benzoyl-4-(hydroxymethyl)piperidin-3-ol
2-amino-6-{4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
9-hydroxy-2-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1-(2,4-dichlorophenyl)-3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
(3S,4S)-1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
N-[2-(2-fluorophenyl)-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl]-N-methyl-3-(methylsulfanyl)propanamide
2-{[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2-(1-methyl-1H-pyrrol-3-yl)-N-(pyridin-3-ylmethyl)acetamide
2-methyl-1-{1-[(2-methyl-1-benzofuran-7-yl)methyl]piperidin-4-yl}propan-1-ol
1-(3-{2-[4-(hydroxymethyl)phenyl]pyridin-4-yl}pyrrolidin-1-yl)-3-(1H-pyrrol-1-yl)propan-1-one
N-[(2R,3R)-2-ethoxy-1'-(thian-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-{2-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine-4-carboxamide
N,N-dimethyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-2-(1H-imidazol-1-yl)ethan-1-one
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,3-oxazole-4-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-5-methyl-1,3-oxazole-4-carboxamide
3-({[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amino}methyl)-N-(pyrazin-2-yl)benzamide
5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
4-(5-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
N-(2-methoxyethyl)-3-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)propanamide
8-methoxy-N-[2-(pyridin-2-ylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{2-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-ethyl-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
2,2-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]oxane-4-carboxamide
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-(5-methylthiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[2-(1H-imidazol-1-yl)ethyl]-3-[(3-methylbutyl)amino]-5-(phenylsulfamoyl)benzamide
1-{1-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
(4aR,7aS)-1-(2-phenylethyl)-4-[2-(1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2-methoxyacetamido)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(4,5-dimethylfuran-2-yl)methyl]piperidine
6-(pyrrolidin-1-ylmethyl)-4-(quinoxalin-2-yl)-1,4-oxazepan-6-ol
1-ethyl-3-[2-(methylsulfanyl)ethyl]-5-(oxan-4-yl)-1H-1,2,4-triazole
(3aR,6aS)-5-[(3-ethoxy-4-methoxyphenyl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[5-(propan-2-yl)-1,2-oxazole-3-amido]cyclopentane-1-carboxylic acid
1-{2-[(1H-indol-7-ylmethyl)(methyl)amino]ethyl}piperidin-2-one
1-ethyl-4-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}piperazin-2-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(morpholin-2-yl)acetamide
(3R,4R)-3-cyclopropyl-1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-4-methylpyrrolidin-3-ol
2-(2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
(4aR,6R,8aS)-2-(furan-2-ylmethyl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
N-(1-ethyl-2-methyl-7-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-5-yl)benzenesulfonamide
N,N-dimethyl-5-{[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1,3-thiazol-2-amine
1-(6-methoxypyrimidin-4-yl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
3-benzoyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
N-[2-(cyclohex-3-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperidin-4-amine
7-(3-chlorophenyl)-4-(2-methylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[2-(azepan-1-yl)ethyl](propan-2-yl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine