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5-chloro-N-[(1S,2R)-2-{[1-(propan-2-yl)piperidin-4-yl]amino}cyclobutyl]thiophene-2-carboxamide
1-{[4-(1H-pyrazol-4-yl)phenyl]methyl}piperazine
N-(2-{1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}ethyl)-2,2-difluoroacetamide
N-butyl-N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-(2-methyl-4-phenylpyridine-3-carbonyl)-4-phenylpiperidin-4-ol
N-cyclopropyl-N-ethyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
(3aR,5R,6S,7aS)-2-(5-fluoro-1H-indole-3-carbonyl)-octahydro-1H-isoindole-5,6-diol
2-[4-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)morpholin-3-yl]-N-(2,2,2-trifluoroethyl)acetamide
(1R,3S)-7-(2,6-difluoro-3-methoxybenzoyl)-7-azaspiro[3.5]nonane-1,3-diol
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(2-methoxyphenyl)-2-methylpiperazine
1-(3-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{[methyl(thian-4-yl)amino]methyl}benzoic acid
N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl (2S)-2-[(1-cycloheptyl-1H-1,2,3-triazol-4-yl)formamido]-3-(4-hydroxyphenyl)propanoate
N-[3-(3-chlorophenyl)phenyl]-1-methanesulfonylpiperidine-4-carboxamide
3-(4-hydroxyphenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
N-(3,5-dimethylphenyl)-2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carboxamide
(3S,4S)-4-methyl-1-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3,4-diol
3-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-(cyclopropylmethyl)-1-methyl-N-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3-carbamoylphenyl)methyl]-N-(4-methoxy-2-methylphenyl)pyrrolidine-1-carboxamide
N2-[2-(azepan-1-yl)ethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(pyridazine-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(naphthalen-2-yl)-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(cyclopropylmethyl)-5-[5-(methoxymethyl)furan-2-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(4-{[4-(aminomethyl)piperidin-1-yl]methyl}phenyl)-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
8-[1-(2-fluorophenyl)cyclopropanecarbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-methyl-3-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridin-2-amine
2-({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}amino)ethan-1-ol
2-tert-butyl-7,7-dimethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-5,6,7,8-tetrahydroquinazolin-5-amine
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
9-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(6-cyanopyridin-3-yl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
1-[(2-methoxyphenyl)methyl]-4-[5-methyl-4-(thiophen-2-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
1-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
4-[3-(4-tert-butylbenzoyl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
4-methyl-2-{1-[1-(propan-2-yl)piperidine-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
4-methoxy-N-[(4-methyl-1,3-thiazol-2-yl)methyl]benzamide
N-(4-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethoxy}phenyl)propanamide
1-[1-(piperidine-1-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-(2-methylphenoxymethyl)piperidine
3-(4-{[2-(dimethylamino)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-en-8-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(2-hydroxybutyl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
5-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
methyl 1-({4-[(1-methyl-1H-pyrazol-4-yl)carbamoyl]phenyl}methyl)piperidine-2-carboxylate
1-[2-({[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
4-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-1λ6-thiomorpholine-1,1-dione
3-[(3R,4S)-1-(5-chloro-3-fluoropyridin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
7-chloro-4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine