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N-(2-chloro-6-methylphenyl)-4-(2,2,2-trifluoroethyl)piperazine-1-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-methyl-1,3-oxazole-4-carboxamide
N-{2-[2-(1H-imidazol-4-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
N-(2-{4-[1-(2-hydroxybutyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)acetamide
5-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1,3-dimethyl-4-[4-(2-methylpropyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(2-methoxyphenyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
8-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(2S)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-hydroxypropanamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-N-(3-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
3-(1-methyl-1H-imidazol-4-yl)-5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazole
N-(2-fluoro-4-methylphenyl)-2-{[4-(methylamino)pyrimidin-2-yl]amino}acetamide
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(thiophen-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclopentyl-3,4-difluoro-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzene-1-sulfonamide
2-[1-(5-fluoro-1-methyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-4-(6-methoxypyridin-2-yl)phenol
2-(4-methoxyphenyl)-N-[(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)methyl]acetamide
(3R,4S)-3,4-dimethyl-1-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-ol
(3aR,5R,6S,7aS)-2-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-octahydro-1H-isoindole-5,6-diol
N-(1-benzylpyrrolidin-3-yl)-3-[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-4-yl]propanamide
1-methyl-2-oxo-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,2-dihydropyridine-3-carboxamide
5-(2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
3-[2-(propylsulfanyl)ethyl]-1-(4-sulfamoylphenyl)urea
2-(2-methoxyethyl)-9-[(3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[9-(2-methoxyethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-2-carbonitrile
1-{3-[({4-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)amino]propyl}pyrrolidin-2-one
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methylthieno[3,2-d]pyrimidin-4-amine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-[(5-cyclopentylthiophen-2-yl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
4-ethyl-N,N-dimethyl-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-2-amine
2-[3-(3-fluorophenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
7-(2-methoxy-5-methylbenzenesulfonyl)-2-methyl-2,7-diazaspiro[4.5]decane
N-[2-(1H-imidazol-4-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(1H-indazol-4-yl)-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
1-[(2-aminopyridin-3-yl)methyl]-4-(3-tert-butyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(3-methylphenyl)methyl]pyrrolidin-3-yl]methanol
2-(dimethylamino)-8-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-chloro-N,N-dimethyl-5-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}-1,3-thiazol-2-amine
2-(3-{[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}phenyl)ethan-1-amine
4-(4,4-difluoropiperidine-1-carbonyl)-1,2-dihydroisoquinolin-1-one
N-{2-[(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazol-4-yl)formamido]ethyl}acetamide
[3-(prop-2-en-1-yl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-3-yl]methanol
5-(propan-2-yl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
8-methoxy-2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}quinoline
N-[2-(3-methoxyphenyl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine