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N-tert-butyl-4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(2-methoxyethyl)-4-[({5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)methyl]pyrrolidin-2-one
methyl 3-[4-({3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)-1H-pyrazol-1-yl]propanoate
1-{1-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidin-3-yl}-3-phenylpropan-1-one
(3R,5S)-N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-(2-methoxy-4-{[(2-phenoxyethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)(quinoxalin-6-ylmethyl)amine
N-(2,4-dimethoxyphenyl)-3-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]propanamide
3-(5-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-{[2-(azepan-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)pent-4-enamide
2-(2-chloro-6-fluorophenyl)-1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]ethan-1-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1,2,3,4-tetrahydronaphthalene-2-carboxamide
2-{2-oxo-2-[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-1,2-dihydrophthalazin-1-one
4-[(3-methylphenyl)sulfanyl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
3-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-[(3S)-2-oxoazepan-3-yl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-(1H-1,3-benzodiazol-1-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
2-(2,6-dimethoxypyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
2-amino-4-[4-(1H-imidazol-1-yl)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1'-(2,3-dihydro-1-benzofuran-2-carbonyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(4-chlorophenyl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}morpholine
3-(3-ethylpiperazine-1-carbonyl)-4-methoxybenzene-1-sulfonamide
1-(2-{[1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)pyrrolidin-2-one
N-butyl-N-(furan-2-ylmethyl)oxolane-2-carboxamide
2-(2-chlorophenyl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
6-cyclopentyl-N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(propan-2-yl)pyrimidine
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-methyl-3-phenylbutan-1-one
N-(thiophen-2-ylmethyl)-1-(2-{[(2,3,4-trimethoxyphenyl)methyl]amino}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-ethyl-2-{6-hydroxy-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,4-diazepan-1-yl}acetamide
methyl 2-{[(2-fluorophenyl)methyl]sulfamoyl}-6-(3-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-cyclopropanecarbonyl-2-(1-methyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-benzyl-5-[1-(2-methoxyphenyl)propan-2-yl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,3S)-7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-azaspiro[3.5]nonane-1,3-diol
1-(4-methoxyphenyl)-6,6-dimethyl-4-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}piperazin-2-one
{[4-({1-[3-(3-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
methyl 2-{[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidine-1-carbonyl]amino}acetate
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
4-chloro-5-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
3-methyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
6-ethyl-N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2-methylquinoline-4-carboxamide
1-(3-methoxyphenyl)-4-[3-(5-methylfuran-2-yl)butyl]piperazin-2-one
1-[1-(2-methylpropyl)piperidin-4-yl]-3-(1H-pyrazol-5-yl)piperidine
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(methanesulfonylmethyl)piperidine
[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-cyclopentyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-(1-benzylpyrrolidin-3-yl)-3-[1-(oxane-4-carbonyl)piperidin-4-yl]propanamide