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N-[2-(piperidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
6-[9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
9-(6-aminopyridine-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)methyl]-1,3-oxazole-4-carboxylate
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
N,2-diethyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}pyrimidine-5-carboxamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}thiophene-3-carboxamide
2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}pyridine-4-carboxamide
N-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
4-ethyl-3-[2-(phenylamino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
3-(4-chlorophenyl)-2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propan-1-ol
2-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2-dihydroquinoline-4-carboxamide
N-{3-oxo-3-[3-(1H-pyrazol-5-yl)piperidin-1-yl]propyl}methanesulfonamide
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
6-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-cyclopentyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-6-oxopiperidine-3-carboxamide
6-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}pyridine-2-carboxylic acid
(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}morpholin-3-yl)methanol
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-(trifluoromethyl)pyridine
2-{5-[1-(2-oxopyrrolidin-1-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl}acetamide
N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-[4-(pyrrolidine-1-sulfonyl)piperazine-1-carbonyl]-1H-1,3-benzodiazole
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
2-(dimethylamino)-7-[4-(1H-pyrazol-4-yl)butanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}pyrrolidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
4-({[(6-chloropyridin-3-yl)methyl](methyl)amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(3-{[1-(2-amino-4-phenylpyrimidine-5-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
1'-(4-ethyl-5-methylthiophene-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(1H-imidazole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-{[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-imidazole
N-(1H-indol-4-ylmethyl)-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-(cyclopropylsulfamoyl)-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]benzamide
(benzylsulfamoyl)(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
5-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N,2-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-sulfamoylbenzamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}propan-1-one
5-(methoxymethyl)-N-[(3R,4S)-1-[2-(methylcarbamoyl)ethyl]-4-(propan-2-yl)pyrrolidin-3-yl]furan-2-carboxamide
1-(2-aminoethyl)-N-[(2-ethoxypyridin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(1,4-dithiepan-6-yl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-ethoxypropan-1-one
2-{3-[(2-phenylazetidin-1-yl)methyl]phenyl}-6-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-(3-benzoylpiperidin-1-yl)-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-5-acetamido-2-hydroxybenzamide
4-[2-methyl-7-(pyrazine-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholine
(1R,6S)-9-methyl-3-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
5-(2-chlorophenyl)-N-[2-(oxan-3-yl)ethyl]furan-2-carboxamide
3-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one
1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}-3-(methoxymethyl)pyrrolidine