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1-[1-(1-benzofuran-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
7-methyl-2-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-2-(pyridin-4-yl)acetamide
8-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}cyclohex-3-ene-1-carboxamide
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-3-(2-phenylphenyl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
1,8-bis(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4,5,6,7-tetrahydro-2H-indazole
(2E)-3-(3-fluorophenyl)-1-[9-(oxan-2-ylmethoxy)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]prop-2-en-1-one
4-{[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}benzamide
1-[(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
5-methoxy-2-{[8-methoxy-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
N-{[4-hydroxy-1-(1,3-thiazol-2-ylmethyl)azepan-4-yl]methyl}benzamide
3-{[3-(methylsulfanyl)propyl]sulfamoyl}-N-(2,2,2-trifluoroethyl)benzamide
3-{2-[3-(2-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
4-(2-methoxyethyl)-3-(1-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-4H-1,2,4-triazole
(3S)-3-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}azepan-2-one
N'-ethyl-N'-[(4-fluorophenyl)methyl]-N-(4-methylphenyl)propanediamide
4-(7-hydroxy-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-N-methylbenzene-1-sulfonamide
N-[(3R,4S)-1-[2-(2,4-dioxoimidazolidin-1-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
1-(2-methoxyphenyl)-3-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-[2-(3-methylphenyl)-1,3-thiazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
4-{7-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholine
N-cyclopropyl-2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}acetamide
8-(1-hydroxypropan-2-yl)-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
7-methyl-2-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
1-(morpholin-4-yl)-3-(1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-4-yl)propan-1-one
(3S,7S,8aS)-7-{[(4-methoxyphenyl)methyl]amino}-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-(furan-3-carbonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-methyl-N-(quinolin-3-ylmethyl)-4-[(thiophen-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
methyl 4-[4-(2,1,3-benzoxadiazol-4-ylmethyl)piperazin-1-yl]benzoate
5-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
6-{3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
2-[(2-amino-6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-yl)amino]ethan-1-ol
2-ethyl-1-(3-methoxypropyl)-7-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-amine
2-(4-methoxyphenoxymethyl)-N-[2-(morpholin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
1'-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
[(2S,6S)-11-methoxy-4-[(4-methoxy-3-methylphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-[(3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1H-pyrazol-5-yl)methyl]-1H-indole
(1R,2R)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-phenylcyclopropane-1-carboxamide
N,N-bis(furan-2-ylmethyl)-N'-(4-methylphenyl)propanediamide
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-[(4-methylpyridin-2-yl)methyl]piperidin-4-amine
(1,3-benzoxazol-2-ylmethyl)({[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl})methylamine
[(3R,4R)-1-(2-ethoxypyridine-3-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}urea
2-{[3-(ethylsulfanyl)propanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide