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N-[(1S,2R)-2-hydroxy-1,2-diphenylethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-methyl-5-{[2-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
6-ethoxy-3-[(4-propylpiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one
5-(2H-1,3-benzodioxol-4-ylmethyl)-2-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-[(isoquinolin-5-yloxy)methyl]-N-[3-(1H-pyrazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
6-methyl-2-({2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}sulfanyl)-3,4-dihydropyrimidin-4-one
2-(dimethylamino)-7-{[2-(prop-2-yn-1-yloxy)phenyl]methyl}-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]-N-(propan-2-yl)acetamide
4-{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrazol-3-yl}benzoic acid
8-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(furan-2-carbonyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
4-ethyl-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(5-fluoropyridine-3-carbonyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
(3aR,7aS)-N-(1H-1,2,3-benzotriazol-5-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
[(4-methoxy-3-methylphenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(diethylamino)-3-[2-methoxy-4-(morpholin-4-ylmethyl)phenoxy]propan-2-ol
4-benzyl-1-(2,3-dihydro-1-benzofuran-7-carbonyl)-3-ethyl-1,4-diazepan-5-one
ethyl 3-[(2-methylphenyl)methyl]-1-(4,4,4-trifluorobutanoyl)piperidine-3-carboxylate
3-benzyl-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]-1,2,4-oxadiazole
1-[(4-methoxyphenyl)methyl]-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2-(methylamino)pyridine-3-carboxamide
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-(propan-2-yl)-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-(3,4-dichlorophenyl)pyrazine
2,4-dimethoxy-N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)benzamide
5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1-benzylpiperidin-3-yl)-5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-{[4-(2-methyl-1,3-benzothiazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-[2-(1-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-2-yl)ethyl]acetamide
(2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-4-yl)methanol
4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
N-(4-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenyl)acetamide
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-(pyrrolidin-1-yl)butan-1-one
ethyl 4-(4-oxo-3,4-dihydroquinazoline-2-carbonyl)piperazine-1-carboxylate
methyl 1-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-4-carboxylate
2-({3-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidine-1-carbonyl]phenyl}amino)acetic acid
1-[4-(2-phenoxyethyl)piperazin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
2-methyl-1-{3-[({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)methyl]piperidin-1-yl}propan-1-one
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-{2-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2-dihydroquinoxalin-2-one
2-(2-hydroxypropyl)-9-[(3-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]amine
2-(2-{1-[2-(2-methyl-1H-indol-3-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-(2-{3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}phenyl)-1,3-diazinane-2,4-dione