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5-fluoro-2-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
2-({[1-(2-methoxyphenyl)ethyl](methyl)amino}methyl)benzonitrile
8-(3-chloro-2-fluorophenyl)-1-methyl-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
N-{[4-(dimethylamino)oxan-4-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-(azepan-1-yl)-N-methyl-4-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-3-phenylpyrrolidin-3-ol
1-cyclopropyl-4-[4-(3,4-difluorobenzoyl)piperidine-1-carbonyl]pyrrolidin-2-one
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
methyl 5-[2-(3-methoxyphenyl)piperidin-1-yl]-5-oxopentanoate
N-methyl-5-phenyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
3-{[1-(5-acetylthiophene-3-carbonyl)pyrrolidin-3-yl]methyl}benzamide
4'-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-benzyl-3-{1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2-chlorophenyl)-3-methyl-N-[3-(propan-2-yloxy)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]pyridin-2-amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N,2,7,8-tetramethylquinoline-4-carboxamide
2-(4-ethoxyphenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
7-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-9H-fluorene-9-carboxamide
(1S,5R)-3-benzyl-6-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
9-[3-(dimethylamino)benzoyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(1-methylpiperidin-4-yl)propanamide
2-{2-[(2-carbamoylmorpholin-4-yl)methyl]-4-(pyridin-2-yl)phenoxy}acetic acid
4-(3-benzyl-1H-pyrazol-5-yl)-1-(oxolane-3-carbonyl)piperidine
6-({[2-(pyridin-2-ylsulfanyl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
2-ethyl-8-[3-(morpholin-4-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[2-(piperazine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
3-butyl-1-methyl-4-[2-(trifluoromethyl)benzoyl]piperazin-2-one
7-(2-phenylethyl)-2-(quinolin-8-ylmethyl)-2,7-diazaspiro[4.5]decane
2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
(1R,5R)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-9-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
4-(5-ethyl-1,3-oxazole-4-carbonyl)-2-(3-phenylpropyl)morpholine
3-[2-(N-methylmethanesulfonamido)ethyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
[4-benzyl-1-(5-methoxy-1H-indole-2-carbonyl)piperidin-4-yl]methanol
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}acetamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(trifluoromethyl)pyrimidin-4-amine
1-ethyl-8-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N7-(2H-1,3-benzodioxol-5-yl)-2,N3,N3-trimethyl-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3,7-dicarboxamide
3-{[4-(dimethylamino)oxan-4-yl]methyl}-1-[4-(1,3-thiazol-4-yl)phenyl]urea
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(2-ethyl-6-methylpyrimidin-4-yl)-4-phenylpiperidine-4-carbonitrile
3-ethyl-1-[3-(4-methoxyphenyl)propanoyl]piperidine-3-carboxylic acid
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]acetic acid
4-amino-N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)pyridine-2-carboxamide
(2S)-2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}-4-methylpentanamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[5-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol