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[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[3-({1-[4-(morpholin-4-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}amine
9-methoxy-3-[(1R,2R)-2-phenylcyclopropanecarbonyl]-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-[(4-fluorophenyl)methyl]-N-(3-hydroxypropyl)-3,4,7-trimethyl-1H-indole-2-carboxamide
2-ethyl-N,4-dimethyl-N-[1-(pyrimidin-4-yl)ethyl]-1,3-oxazole-5-carboxamide
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-5-methoxy-4H-pyran-4-one
5-chloro-4-{[4-(2,6-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,3-dimethyl-1H-pyrazole
3-cyclopentyl-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-3-(thiophen-3-ylmethyl)urea
(1S,5R)-6-[(5-chlorothiophen-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,3R)-3-benzenesulfonamido-N-(furan-3-ylmethyl)-N-methylcyclopentane-1-carboxamide
3-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)benzonitrile
4-benzyl-1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-2-one
4-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
N-cyclopropyl-1-[1-(9H-purin-6-yl)piperidin-4-yl]piperidine-4-carboxamide
N-[(2R,4R,6S)-2-cyclohexyl-6-{pyrazolo[1,5-a]pyrimidin-3-yl}oxan-4-yl]acetamide
N-[2-(4-methoxyphenyl)ethyl]-2-(trifluoromethyl)morpholine-4-carboxamide
8-(6-aminopyrimidin-4-yl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(3-methoxybenzoyl)-1-(1,2-oxazol-3-ylmethyl)piperidine
5-{[(4aS,7aR)-6,6-dioxo-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-1-methyl-1H-indole
2-(2,4-difluorophenoxy)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]acetamide
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
2-[1-(4-methyl-3-phenyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]benzoic acid
4-{[1-benzyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
1-{3,5-dimethyl-4-[4-(pyridin-4-yl)-1,4-diazepane-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
N-[3-(4-ethylpiperazin-1-yl)propyl]-4-(piperidin-3-yl)benzamide
7-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-2-methyl-2,7-diazaspiro[4.5]decane
3-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-N-[(4-fluorophenyl)methyl]propanamide
2-{2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-indazol-3-one
ethyl 1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
7-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(2-methyl-5-propylpyrimidin-4-yl)-N-{1-oxaspiro[4.5]decan-3-yl}piperidin-4-amine
4-(2H-1,3-benzodioxol-5-yloxy)-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
4-(2-{4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
2-(2-chlorophenoxy)-N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(5-methylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methoxypyridine-4-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(4-ethylpiperazin-1-yl)ethan-1-one
2-amino-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-1H-pyrrole-2-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide
1-cyclopentanecarbonyl-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-cyclopentyl-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-2-one
1-ethyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1H-pyrazole-5-carboxamide
(1S,6R)-9-(1,4-dithiepan-6-yl)-3,9-diazabicyclo[4.2.1]nonane
3-(1H-pyrazol-4-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
N-[(2-chlorophenyl)methyl]-3-[1-(1-phenylpiperidin-4-yl)piperidin-3-yl]propanamide
4-cyclopropyl-6-[3-(2-methoxyphenoxy)azetidin-1-yl]pyrimidine
ethyl 3-benzyl-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-3-carboxylate