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6-fluoro-2-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}quinolin-4-ol
5-({[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]amino}methyl)-N-methylfuran-2-carboxamide
2-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
methyl 4-[4-(2-methoxypyridine-4-carbonyl)piperazin-1-yl]benzoate
(4aS,7aR)-1-(3-acetyl-1H-pyrazole-5-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-({3-[(4-chlorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-ethyl-1H-1,2,4-triazole
3-(aminomethyl)-4-(5-chloro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-benzofuran-2-ylmethyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
2-(1-ethylpiperidin-4-yl)-1-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]ethan-1-one
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]thiophene-3-carboxamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[3-(1H-imidazol-1-yl)propyl]propanamide
1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
9-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
5-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrazin-2-ol
N-benzyl-4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-sulfonamide
1-(2-methoxyethyl)-3-(2-methylpropyl)-8-(oxan-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(3R,4R)-1-(3-chloro-4-methylbenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propan-1-one
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2,2-dimethylpropan-1-one
methyl[2-(pyridin-4-yl)ethyl]{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}amine
2-cyclopropyl-8-(9H-purin-6-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-N-phenylpyrimidin-2-amine
4-({4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
2-[2-(1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1H-imidazol-2-yl)phenoxy]acetic acid
2-ethyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-4-methyl-1H-imidazole
4-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
3-(1-methyl-1H-pyrazol-4-yl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]propanamide
5-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-2-ol
N-(1-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
1-(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
1-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-3-{2-methylimidazo[1,2-a]pyridin-5-yl}urea
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-3-(quinolin-8-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-(2-chlorophenyl)-2-(4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-[(isoquinolin-5-yloxy)methyl]-N-[1-(1-methylpiperidin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
4-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidine-1-carbonyl)pyridine
1-{3-[4-(1-ethoxyethyl)phenyl]phenyl}piperazine
(1R,5R)-N,N-dimethyl-6-[3-(5-methylfuran-2-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
6-[(diethylamino)methyl]-N-(2,3-dihydroxypropyl)-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S,4S)-1-benzyl-N-(pyridin-3-ylmethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
{[5-(3-chlorophenyl)furan-2-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
5-chloro-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
(3S,4R)-1-[(2-amino-4-chloro-1,3-thiazol-5-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
5-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
(3S,4R)-N-cyclohexyl-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carboxamide
1-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-1H-indole-3-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
1-(4,7-dimethylquinazolin-2-yl)-N-(2-phenylethyl)azepan-4-amine
4-(3-chloro-4-fluorophenyl)-1-[2-(propane-2-sulfonyl)ethyl]-1H-1,2,3-triazole
2-(4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)ethan-1-ol