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(3R,4S)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-cyclopropylpyrrolidin-3-amine
2-({[(3R,4R)-1-(5,6-dimethylpyridine-3-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-amino-6-(2,5-dimethylphenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
4-(piperidin-1-yl)-1-(1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidine-4-carboxamide
2-[2-amino-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]pyridine-3-carbonitrile
1-(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
1-cyclopentyl-4-[4-(2,4-difluorophenyl)-5-methyl-1H-imidazol-2-yl]pyrrolidin-2-one
7-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(propan-2-yl)-1-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
(3aR,6aR)-2-(5-cyano-4,6-dimethylpyridin-2-yl)-5-cyclohexyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-(piperidin-1-yl)piperidine-1,4-dicarboxamide
1-(4-methyl-1,4-diazepan-1-yl)-3-(2-methylphenyl)-3-phenylpropan-1-one
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
N-[2-(3-fluorophenyl)ethyl]-2-(4-{4-[(1,3-thiazol-2-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
6-[2-(4-methylbenzenesulfonyl)ethyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
3-methyl-2-oxo-N-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
4-hydroxy-N-methyl-N-{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
3-(3-methoxypropyl)-1-[2-(methylsulfanyl)acetyl]piperidine-3-carboxylic acid
N-(3-ethoxypropyl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4S)-1-[2-(2-aminoethyl)quinazolin-4-yl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-5-(methoxymethyl)furan-2-carboxamide
[(3R,4R)-1-[4-(furan-2-yl)benzoyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
5-oxo-N-[3-(trifluoromethyl)phenyl]-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
4-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperazin-2-one
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-4-methylpyrimidine-5-carboxamide
8-[(4-carboxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[1-benzyl-3-(3-oxopiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N,N-diethylacetamide
1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(4S)-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4-phenyl-1,3-oxazolidin-2-one
4-({2-[3-(morpholin-4-yl)propoxy]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
2-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)-5-fluoro-1H-1,3-benzodiazole
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
1-(1-methylpiperidin-4-yl)-4-[4-(pyrrolidin-1-yl)benzoyl]piperazine
N-(cyclohexylmethyl)-6-(2,5-dimethoxyphenyl)-2-(4-methylpiperazin-1-yl)pyridine-3-carboxamide
3-[(3R,4S)-1-(5-fluoro-2-methoxybenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
5-(hydroxymethyl)-2-methyl-4-{[methyl({[3-(methylsulfanyl)phenyl]methyl})amino]methyl}pyridin-3-ol
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(furan-3-carbonyl)-1,4-diazepan-6-ol
8-[(3-ethenylphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(oxan-4-yl)-1,4-diazepan-6-ol
(3R,4R)-1-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3,4-dimethylpyrrolidin-3-ol
3-{pyrazolo[1,5-a]pyridin-7-yl}-6-(pyrrolidin-1-yl)pyridazine
4-hydroxy-N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-phenylpyrimidine-5-carboxamide
2-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]thiophene-3-sulfonamide
5-[4-(1-benzylpyrrolidin-3-yl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
3-(4-fluorophenyl)-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
2-methyl-6-[(thiolan-3-yl)amino]heptan-2-ol