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4-[(2-methyl-1H-imidazol-1-yl)methyl]-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperidine-1-carboxamide
[2-(1H-imidazol-1-yl)ethyl]({[7-methoxy-2-(thiophen-3-yl)quinolin-3-yl]methyl})amine
2,4-difluoro-N-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
(4aS,8aR)-6-{2-[4-(hydroxymethyl)phenyl]acetyl}-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
1-[(3-fluorophenyl)methyl]-4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]acetic acid
2-[(4-chlorophenyl)sulfanyl]-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-[(3S,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1-(propan-2-yl)-1H-pyrrole-2-carboxamide
N-methyl-5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrimidin-2-amine
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-phenylethane-1,2-dione
N-cyclopentyl-1-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
7-methoxy-3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-[1-(3,5-dimethylphenyl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
ethyl 4-[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]piperidine-1-carboxylate
methyl 5-oxo-5-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]pentanoate
N3-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)propane-1,3-diamine
(3R)-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
7-methyl-2-(5-propyl-1,3,4-oxadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-thiazole-5-carboxamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
2-({2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
2-(methylsulfanyl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-1,3-thiazole-4-carboxamide
1-[(5-ethylpyridin-2-yl)methyl]-4-(pyridin-4-yl)piperazine
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-4-methoxy-3,5-dimethylbenzamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(propylsulfanyl)acetyl]pyrrolidin-3-yl]acetamide
2-(4-{[(2-ethylphenyl)carbamoyl]formamido}-3,5-dimethyl-1H-pyrazol-1-yl)acetic acid
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5S,9aS,9bS)-5-(4-hydroxy-3,5-dimethylphenyl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2-methyl-1,4-dihydropyridin-4-one
5-{thieno[3,2-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)benzonitrile
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(3-phenylpropanoyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-[3-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
2-[1-(1,3-benzothiazol-2-yl)-1,4-diazepan-6-yl]acetic acid
(2S,4R)-N-ethyl-1-(furan-2-carbonyl)-4-[2-(pyrazin-2-yl)acetamido]pyrrolidine-2-carboxamide
5-methyl-4-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}pyrimidin-2-amine
4-{3-[(4-hydroxyphenyl)methyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl}benzoic acid
2-[2-methyl-4-(quinolin-8-yl)phenoxy]acetamide
2-amino-1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
4-chloro-5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
1-(4-ethenylphenyl)-3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}urea
2-[4-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
[(4aS,8aR)-6-{furo[3,2-c]pyridin-4-yl}-decahydro-1,6-naphthyridin-4a-yl]methanol
3-(1-benzofuran-2-yl)-4-{1H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
7-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
4-benzyl-3-ethyl-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1,4-diazepan-5-one
6-methyl-5-{5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[(2-chlorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methyl-5-({4-phenyl-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1H-imidazol-1-yl}methyl)pyrazine
6-amino-N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]pyridine-3-carboxamide