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(3R,4S)-4-cyclopropyl-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-N,N-dimethylpyrrolidin-3-amine
5-[5-(methoxymethyl)-3-methyl-1H-pyrazol-4-yl]-8-methylquinoline
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
N-cyclohexyl-3-(5-methylfuran-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(1H-pyrazol-1-yl)acetamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3-fluorophenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
5-methoxy-1-methyl-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H-indole-2-carboxamide
4-methyl-6-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]pyrimidin-2-amine
7-fluoro-3-methyl-2-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carboxamide
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-4-oxo-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(1-ethylpiperidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
8-[2-(2-chloro-4-fluorophenyl)acetyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-(3-propyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methoxy-N-methylpyridine-3-carboxamide
(1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
5-chloro-2-methoxy-4-(1-propyl-1H-1,2,4-triazol-5-yl)pyridine
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-[(5-methylfuran-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
[(3R,4R)-1-{[2-(methylsulfanyl)phenyl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
6-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-ylmethyl]pyridine-2-carboxylic acid
8-(2-aminopyridine-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(prop-2-en-1-yl)-N-[2-(propan-2-yloxy)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4-(thiophen-2-yl)butanamide
3-({3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
1-[2-(dimethylamino)-4-[2-(2-methoxyethyl)morpholin-4-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}piperidin-3-ol
N-(cyclohexylmethyl)-2-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]acetamide
(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
(1S,5R)-3-{[3-(2-aminoethyl)phenyl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(adamantan-2-yl)-2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-[methyl(piperidin-4-yl)amino]ethan-1-one
(3S,5R)-1-(4-ethyl-5-methylthiophene-3-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
3-(2-methylpropyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1,2-oxazole-5-carboxamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-3-(3-methoxyquinoxalin-2-yl)propan-1-one
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
1-({5-hexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-({4-methyl-5-[1-(oxan-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-[3-(methylcarbamoyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2,5-dihydro-1H-pyrrole-2-carboxamide
2-{6-[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
N-ethyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
(3S,4S)-1-[(4-methanesulfonylphenyl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-(6-cyanopyridin-3-yl)-3-[(diethylamino)methyl]benzamide
5-[2-(adamantan-1-yl)acetyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
2-(pyrimidin-2-ylsulfanyl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide