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1-{1-[3-(pyridin-3-yl)propyl]piperidin-4-yl}propan-1-ol
N-[1-(2-methoxyphenyl)propan-2-yl]-N-methyl-4-propylpyrimidine-5-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(3-propyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
2-(4-acetylpiperazine-1-carbonyl)-3,4-dihydroquinazolin-4-one
3-chloro-N-(2-methoxyethyl)-4-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
3-{[(2,2-difluoroethyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]methyl}-1,3-oxazolidin-2-one
4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
2-ethoxy-1-[(3S,4S)-3-hydroxy-4-[4-(2-methoxyphenyl)piperazin-1-yl]pyrrolidin-1-yl]ethan-1-one
2-[(3-propoxypiperidin-1-yl)methyl]benzoic acid
N-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-sulfonamide
8-{3-cyclopropyl-5-[(pyridin-3-yloxy)methyl]-1H-1,2,4-triazol-1-yl}quinoline
2-[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-N-(2-methoxy-5-methylphenyl)acetamide
ethyl 3-{[7-(2-chlorobenzamido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]amino}propanoate
N-(furan-2-ylmethyl)-3-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propanamide
5-(2-{2-[(6-cyclopropylpyrimidin-4-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]acetamide
2-(3-methylbutanoyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(5-{1-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1H-imidazol-2-yl}furan-2-yl)methanol
1-{4-[cyclopentyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]piperidin-1-yl}ethan-1-one
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
N-ethyl-2-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-benzoxazole-6-carboxamide
(4aS,7aR)-1-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-6-[3-(methoxymethyl)piperidin-1-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N-(butan-2-yl)-3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]benzamide
7-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
N-ethyl-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]pyrimidin-2-amine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-[(3aR,6aR)-2-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-2,5-dihydro-1H-pyrrole
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-thiazole-5-carboxamide
5-(2,4-difluorophenoxymethyl)-N-(2-oxopiperidin-3-yl)-1H-pyrazole-3-carboxamide
2,5,6-trimethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrimidin-4-amine
{3-benzyl-1-[3-(2-fluorophenyl)benzoyl]piperidin-3-yl}methanol
N-{2-[2-(1H-indol-3-yl)acetamido]-4-methylphenyl}pentanamide
1-(4-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}thiophen-2-yl)ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(4-ethylpiperazin-1-yl)-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-[4-(piperidine-1-carbonyl)phenyl]urea
4-(piperidin-3-ylmethyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]benzamide
(1S,5R)-3-{4-[(2-fluorophenyl)methoxy]benzoyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-6-methyl-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
methyl 2-(tert-butylsulfamoyl)-6-{[2-(trifluoromethyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3,4-dimethylphenoxy)ethan-1-one
2,6-dimethyl-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrimidine-4-carboxamide
{imidazo[1,2-a]pyridin-3-ylmethyl}({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine