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4-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
(2S,4S)-4-amino-N-ethyl-1-[2-(methylamino)pyridine-3-carbonyl]pyrrolidine-2-carboxamide
N-[(3R,4S)-1-(2-aminopyrimidin-4-yl)-4-propylpyrrolidin-3-yl]-3-methoxypropanamide
N-cyclopentyl-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
3-(pentan-2-yl)-8-(1-propyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4S)-4-amino-1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-N,N-diethylpyrrolidine-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1,3-dimethyl-N-[3-(4-methylpiperazin-1-yl)butyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2S,4R)-4-amino-N-ethyl-1-[2-(trifluoromethyl)benzenesulfonyl]pyrrolidine-2-carboxamide
2-{2-[(4,4-difluoropiperidin-1-yl)methyl]-6-methoxyphenoxy}propanoic acid
6-ethyl-N4-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N2,N2-dimethylpyrimidine-2,4-diamine
2-ethoxy-6-{[4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenol
1-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(1-ethyl-2-methyl-1H-indol-5-yl)urea
1-(2-methylpropyl)-N-(naphthalen-1-ylmethyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
6-ethyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]pyrimidin-4-amine
3-{[(butan-2-yl)(cyclopentyl)amino]methyl}-7-fluoro-1,2-dihydroquinolin-2-one
3-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-imidazol-2-yl}pyridine
methyl[(3-methylquinoxalin-2-yl)methyl]{[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-(4-fluorophenoxy)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
4-(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1,3-thiazol-2-yl)morpholine
1-[3-(azocan-1-yl)propanoyl]piperidine-4-carboxylic acid
N-[(3R,4S)-4-cyclopropyl-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl]methanesulfonamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(3-methoxyphenyl)ethan-1-one
(2R,4S)-4-hydroxy-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidine-2-carboxylic acid
N-(cyclopropylmethyl)-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-(2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)cyclopentan-1-ol
8-chloro-2-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}quinolin-4-ol
N-(2-chlorophenyl)-4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
3-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
3-hydroxy-1-(2-methoxyethyl)-3-({[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)piperidin-2-one
2-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxypyridin-4-ol
2-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-3,4-dimethoxypyridine
4-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}-1,4-oxazepane
N'-(2-ethoxyphenyl)-N-[2-(2-hydroxyethoxy)ethyl]propanediamide
2-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1-methylazepane
1-[(2,5-dimethoxyphenyl)methyl]-3-(1-propyl-1H-1,2,4-triazol-3-yl)urea
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(4-methoxyphenyl)ethyl]methylamine
(3S,4S)-1-[3-(difluoromethoxy)benzoyl]-4-methylpiperidine-3,4-diol
(3S,4R)-4-(2-methoxyphenyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-3-carboxylic acid
5-(2-methyl-5-propylpyrimidin-4-yl)thiophene-2-carboxylic acid
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine
4-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-1-(oxolane-2-carbonyl)piperidine
5-({2-[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}methyl)-N-methylfuran-2-carboxamide
1-(2-{[(2-chlorophenyl)methyl](methyl)amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
4-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(3S)-3-(dimethylamino)azepan-1-yl]-5-phenylpentane-1,5-dione
N-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-methyl-2-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
(1R,3S)-3-(2-aminoethoxy)-7-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-7-azaspiro[3.5]nonan-1-ol