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1,5-dimethyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-3-carboxamide
ethyl 4-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)-1H-pyrazole-3-carboxylate
6-fluoro-4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(3-fluorophenoxy)piperidine
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
3,3-dimethyl-1-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}urea
(3aS,6aS)-1-oxo-5-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[7-oxo-5-(4-propylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]thiophene-2-carboxamide
2-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-3-ethyl-1H-indole
4-[3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-8-methylquinolin-2-yl]piperazin-2-one
N-[2-(propylsulfanyl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
9-(cyclohex-3-en-1-ylmethyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-4-fluoropiperidine
3-({[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl](cyclopropyl)amino}methyl)phenol
2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]acetamide
4-(azonan-1-yl)-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
(3S,4R)-1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}-4-phenylpyrrolidine-3-carboxylic acid
2-(3-fluorophenoxymethyl)-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
(dicyclopropylmethyl)(methyl){[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-methylpiperazin-2-yl]ethan-1-ol
1-[2-methoxy-4-({[3-(2-methyl-1H-imidazol-1-yl)propyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
1-(4-fluorophenyl)-4-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}piperazine
4-[(diethylamino)methyl]-5-ethyl-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]furan-2-carboxamide
1-methyl-4-{2-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]ethyl}piperidin-4-ol
2,5-dimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-(oxan-3-yl)pyrimidin-2-amine
N-cyclopropyl-2-[3-(2-ethylphenoxy)azetidin-1-yl]pyridine-4-carboxamide
(2S)-2-amino-N-ethyl-3-methoxy-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
N-[(3-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-[1-(ethylcarbamoyl)piperidin-4-yl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
7-chloro-3-({[(2-methoxyphenyl)methyl]amino}methyl)-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
({4-ethyl-5-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-ethyl-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-4-methyl-1,3-oxazole-5-carboxamide
methyl 6-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(3-methylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[2-(1H-pyrazol-1-yl)ethyl]pyridin-2-amine
4-({2-[6-(propan-2-yloxy)pyridazin-3-yl]phenyl}methyl)morpholine
N-methyl-2-{3-[3-(quinoxalin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-cyclohexyl-3-[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
6-(azepan-1-yl)-N-(oxolan-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(3aR,6aR)-2-cyclobutanecarbonyl-5-(2,3-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
[(3R,4R)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(5-chloropyridin-2-yl)-4-[(1-ethylpiperidin-2-yl)methyl]piperazine
1-methyl-N-[(6-methylpyridin-2-yl)methyl]-N-(2-phenylethyl)piperidin-4-amine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]acetamide
3-(3,4-difluorophenyl)-5-(3-ethynylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(ethyl)(oxan-4-ylmethyl)amine