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3-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
N2-(2-methoxyethyl)-N4-methyl-N4-[(5-methyl-1H-pyrazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(2,2-dimethyloxan-4-yl)-N-ethyl-1-(methoxymethyl)cyclobutane-1-carboxamide
1-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-6-ol
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(1H-indole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[4-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]acetamide
1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-5-yl)urea
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]methanol
2-(dimethylamino)-2-(4-fluorophenyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1,2,3,4-tetrahydroquinolin-2-one
4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-2-(2-methoxyethyl)morpholine
2-{5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
8-(4-chlorobenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
5-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-[4-({ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-2-methylbut-3-yn-2-ol
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-cyclopentylpiperidin-2-one
1-(2-benzyl-1,3-thiazole-4-carbonyl)-3,4,4-trimethylpyrrolidin-3-ol
3-ethyl-1-[3-(furan-2-yl)phenyl]-3-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}urea
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]pyrrolidine-3-carboxylic acid
2-{2-[(dimethylamino)methyl]phenoxy}-4,6-dimethylpyridine-3-carbonitrile
N-(1,3-benzothiazol-2-ylmethyl)-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-methylacetamide
6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
2-methyl-5-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
4-methyl-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]-3-(2-oxoimidazolidin-1-yl)benzamide
2-methyl-N-[2-({4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-6-yl}amino)ethyl]propanamide
1-(2,4-dimethylphenyl)-3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}urea
2-(3-methylbut-2-en-1-yl)-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
ethyl 3-(3-phenylpropyl)-1-(pyrazine-2-carbonyl)piperidine-3-carboxylate
1-methyl-N-(2-phenylethyl)-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-chlorophenyl (7S,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(5-{1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
1-{2-[5-(5-methyl-4,5,6,7-tetrahydro-2H-indazol-3-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
(1S,5R)-6-(2,3-dimethyl-1H-indole-7-carbonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-(3-methoxypropyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-phenylpropanamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)piperidine-1-carboxamide
2,5-dimethyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[(2S)-pyrrolidin-2-ylmethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[5-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
3-(1H-pyrazol-1-ylmethyl)-N-(thiophen-3-ylmethyl)benzamide
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
5-amino-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1H-pyrazole-3-carboxamide
6-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3-dihydropyridazin-3-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
1-[(2,6-difluoro-3-methylphenyl)methyl]-4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazole
4-(3-phenylpropyl)-N-(trimethyl-1H-pyrazol-4-yl)-1,4-diazepane-1-carboxamide
6-(piperidin-3-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]pyrimidin-4-amine
1-methyl-4-[5-(naphthalen-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]piperidine
5-fluoro-2-[4-(pyridin-4-yl)piperazin-1-yl]pyrimidin-4-ol