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(2S)-N-cyclohexyl-2-acetamido-N-[2-(ethylsulfanyl)ethyl]-3-(1H-imidazol-4-yl)propanamide
4-(3-cyclohexyl-1H-pyrazol-4-yl)-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-methyl-4-({4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]-2-{[2-(pyridin-2-yl)ethyl]amino}acetamide
methyl 3-acetamido-5-[(4-hydroxybutan-2-yl)amino]-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(dimethyl-1,3-thiazole-5-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
2-ethyl-8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{[(2S)-1-methoxy-3-methyl-1-oxobutan-2-yl]carbamoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
4-(4-methyl-1H-pyrazol-3-yl)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidine
2-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]pyridazine-3-carboxamide
N-[(2S)-4-methyl-1-oxo-1-(3-oxo-4-phenylpiperazin-1-yl)pentan-2-yl]acetamide
1-(2-methoxy-6-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
[1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)pyrrolidin-3-yl]methanol
2-(2-methyl-1,3-thiazol-4-yl)-1-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)ethan-1-one
[(2S,6S)-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
4-[4-ethyl-6-(5-fluoro-2-methoxyphenyl)pyrimidin-2-yl]morpholine
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
7-(cyclobutylmethyl)-2-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-benzothiazole-6-carboxamide
1-methyl-3-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
11-(cyclopropylamino)-4-[(4-methylphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[4-(piperidin-1-yl)benzoyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)butanamide
N,1-dimethyl-N-[(1-methylpiperidin-2-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(1H-imidazol-1-ylmethyl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-ol
2-(2-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}ethyl)pyridine
2-[2-(pyridin-4-yl)ethyl]-9-[2-(pyrrolidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)[(2-ethylpyrimidin-4-yl)methyl]methylamine
N-[(2-ethoxypyridin-3-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
4-(2-ethoxyphenyl)-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-(difluoromethyl)-1H-pyrazole-5-carboxamide
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxy-2-methylpropan-1-one
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-[2-(pyridin-3-yl)ethyl]propanamide
3-(4-fluorophenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
4-{3-[(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)oxy]benzoyl}morpholine
2-[(2-chlorophenyl)methyl]-4-(pyrrolidine-1-sulfonyl)morpholine
2-{3-cyclopropyl-5-[2-methyl-5-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-1-yl}acetic acid
methyl 2-hydroxy-5-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)benzoate
2-methoxy-6-[2-(pyridin-2-yl)ethyl]-3-{[(pyrimidin-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
8-{[3-(2-aminoethyl)phenyl]methyl}-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[2,5-dioxo-4-(piperidin-4-yl)-4-propylimidazolidin-1-yl]methyl}-N-methylfuran-2-carboxamide
N-[(2-methoxyphenyl)methyl]-1,3-dimethyl-N-(2-methylpropyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-amino-4-ethyl-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3-thiazole-5-carboxamide
3-{[4-(dimethylamino)oxan-4-yl]methyl}-1-[3-(methylsulfanyl)phenyl]urea
1-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propane-1,2-dione
1-{2-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyrimidin-2-one
2-{2-[4-(2-fluorophenoxy)piperidin-1-yl]ethyl}-2H-indazole