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2-(1-benzylpiperidin-4-yl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,3-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[2-(2-fluorophenyl)-1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)ethyl]-N-methylthiophene-3-carboxamide
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
4-ethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}benzamide
2-[3-({[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]carbamoyl}amino)phenyl]-N-methylacetamide
3-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2-methylphenol
ethyl 1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-(2,6-dimethoxyphenyl)-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
2-[4-(1-cyano-1-methylethyl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
N-ethyl-2-{4-[(2R)-2-hydroxy-2-(naphthalen-2-yl)acetyl]piperazin-1-yl}acetamide
4-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-(2,3-dihydro-1H-inden-2-yl)-N,2-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(1H-1,2,3-benzotriazol-5-yl)-3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]urea
methyl 5-cyano-6-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-methylpyridine-3-carboxylate
3-[(3R,4S)-3-[3-(4-chloro-1H-pyrazol-1-yl)propanamido]-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
2-{1-[(4-ethoxyphenyl)methyl]-4-[(5-ethylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[(4-methylphenyl)amino]-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-2-phenylpropanamide
7-(cyclopropanesulfonyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
3-(3-methoxyphenyl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
1-[(1-{6-[(furan-2-ylmethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(2E)-3-(3-chlorophenyl)-1-(3-{[(dimethylsulfamoyl)amino]methyl}piperidin-1-yl)prop-2-en-1-one
3-{5-butyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-6-methoxyquinolin-2-ol
(1-{1-[(3-chlorothiophen-2-yl)methyl]piperidin-4-yl}piperidin-3-yl)methanol
5-{3-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-ethylpyrrolidin-2-one
3-{2-oxo-2-[4-(pyridin-4-yl)piperazin-1-yl]ethyl}-4-(2-phenylethyl)piperazin-2-one
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(6-methoxypyrimidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 6-{[benzyl(methyl)amino]methyl}-3-(2-chlorobenzamido)thieno[2,3-b]pyridine-2-carboxylate
ethyl 1-(tert-butylcarbamoyl)-3-[(3-chlorophenyl)methyl]piperidine-3-carboxylate
N,1-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-{[1-butyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-2H-indazole
N-(1-{7-[(2-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
6-({[2-(5-methylfuran-2-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
N-[(2S,4R,6S)-2-benzyl-6-(pyridin-4-yl)oxan-4-yl]benzamide
N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)pent-4-ynamide
1-{2-[(3-methylpyridin-2-yl)amino]ethyl}-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
5-[1-(furan-2-ylmethyl)pyrrolidin-2-yl]-N-(1H-imidazol-2-ylmethyl)thiophene-2-carboxamide
4-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
10-methoxy-5-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-(4-ethylphenyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}-1-(furan-3-carbonyl)piperidine
N-[2-(furan-2-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-[1-(2-benzyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]pyridine
(3R,4S)-4-cyclopropyl-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrrolidin-3-amine
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
2-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
7-(1-benzothiophen-3-yl)-4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol