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2-tert-butyl-4-hydroxy-N-{[4-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
1-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-3,3-dimethylurea
3-{5-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-(3-aminothiophene-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-oxoethyl)-7-methoxy-4-methyl-2H-chromen-2-one
(3aR,5R,6S,7aS)-2-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydro-1H-isoindole-5,6-diol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(1-methyl-1H-pyrazol-4-yl)pyridine
6-{1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}pyrimidin-4-ol
1-{4-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]phenyl}piperidine
N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(propan-2-yl)piperidine-3-carboxamide
1-[(3aS,6aS)-1-cyclopropanecarbonyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-[2-(methylsulfanyl)phenyl]-2-(3-oxopiperazin-1-yl)acetic acid
1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-N-phenylpiperidin-3-amine
ethyl 3-benzyl-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
4-[(3S)-3-ethylmorpholine-4-carbonyl]-N-methylpyridin-2-amine
1-{1-[6-(isoquinolin-5-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
8-[3-(1H-pyrazol-1-yl)propyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
2-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}-6-methylpyridin-3-ol
1-{1-[4-(3-methoxyphenyl)phenyl]piperidin-4-yl}piperidine-4-carboxamide
[(5-chloro-2,3-dimethoxyphenyl)methyl](methyl)[(3-methyl-1H-pyrazol-4-yl)methyl]amine
1-[(4-methanesulfonylphenyl)methyl]-2-(methoxymethyl)piperidine
3-(3-chlorophenyl)-N-(1-hydroxy-2-methylpropan-2-yl)-3-phenylpropanamide
2-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]benzoic acid
N-(2-methoxyethyl)-3-(1H-pyrazol-1-yl)benzamide
5-ethyl-N4-methyl-N4-[(3-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
5-ethyl-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-methylthieno[2,3-d]pyrimidin-4-amine
2-[4-methyl-6-({[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}amino)pyrimidin-2-yl]phenol
5-(cyclopropylmethyl)-2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
methyl 6-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine-4-carboxylate
4-(1-benzofuran-5-yl)-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-amino-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}pyrrolidine-3-carboxylic acid
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(methylamino)-N-[3-(4-methylbenzenesulfonamido)propyl]pyrimidine-5-carboxamide
N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-butyl-5-(1H-pyrazol-3-yl)furan-2-carboxamide
[(4-fluoro-3-methoxyphenyl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine
(2R,3S,6R)-5-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(5-methoxyfuran-2-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
N3-methyl-N5-[1-(naphthalen-1-yl)ethyl]-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}acetamide
5-fluoro-2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3,8-dimethylquinoline
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-cyclopropyl-4-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
9-(3,5-difluoropyridine-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole