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5-fluoro-2-(4-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyrimidine
5,6-dimethyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-(4-cyano-2-ethylphenyl)-3-{[3-(hydroxymethyl)piperidin-1-yl]methyl}benzamide
5-(propan-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
(4aS,7aR)-1-[2-(2,5-dimethylphenyl)acetyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{2-benzyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}benzonitrile
3-[(4-methoxyphenyl)methyl]-1-methyl-8-{[4-(methylsulfanyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-4-phenoxy-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
N-(furan-3-ylmethyl)-2-methyl-1-benzofuran-5-carboxamide
7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-(cyclopropylmethyl)-2-[2-(pyrimidin-2-ylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2-fluorobenzoyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
4-(2-chloro-4-fluorophenyl)-7-(2-methoxyethoxy)-1,2,3,4-tetrahydroquinolin-2-one
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(furan-2-yl)-2-oxoacetamide
2-[2-(6-methylpyridin-2-yl)ethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(oxan-4-yl)ethyl]benzamide
3-(4-chlorophenyl)-3-phenyl-N-[(1r,4r)-4-hydroxycyclohexyl]propanamide
{4-[2-amino-7-methyl-4-(3-methylphenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}methanol
N,1,3-trimethyl-N-(oxan-2-ylmethyl)-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-cyclopropyl-N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-pyrazole-5-carboxamide
1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-4-yl)ethan-1-one
N-[(2-fluorophenyl)methyl]-4-{4-[methyl(oxan-4-yl)amino]piperidin-1-yl}benzamide
1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4-methyl-1,2,3,6-tetrahydropyridine
N-[(1-ethyl-1H-indazol-3-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
1-[(2,6-difluorophenyl)methyl]-N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
2-[2-(3-methoxyphenyl)ethyl]-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-[5-(3,5-difluoro-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]butan-2-ol
1-ethyl-5-(2-propylpyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-benzyl-1-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-cyclohexyl-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]piperidine-4-carboxamide
(cyclohex-3-en-1-ylmethyl)({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
5-chloro-3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-(4-{[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)acetic acid
2-(2-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
2-{1-cyclopentyl-4-[(5-ethylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-methoxy-1-methyl-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-1H-indole-2-carboxamide
1-(3-methyl-3-phenylbutanamido)cycloheptane-1-carboxamide
1-(4-{[(3-methylpyridin-2-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
(5-{1-[(5-methoxy-1H-indol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
3-benzyl-5-(oxolan-2-yl)-1,2,4-oxadiazole
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[(2S)-pyrrolidin-2-ylmethyl]piperidin-4-amine
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[1'-(1-ethylpyrrolidine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
7-[2-(4-methoxyphenoxy)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
11-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one