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N-(morpholin-2-ylmethyl)-4-propylpyrimidine-5-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}propanamide
4-(3,5-dimethoxyphenyl)-6-methyl-5-(1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2,3,4-tetrahydropyrimidin-2-one
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
N-cyclohexyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
5-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-benzyl-1H-1,2,4-triazole
1-[4-(2-methylphenoxy)piperidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
2-[(3-methoxyphenyl)amino]-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}butanamide
2-amino-1-[2-(4-fluorophenyl)piperidin-1-yl]ethan-1-one
(2-{8-[(2-methoxyethyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}-2-oxoethyl)urea
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 4-{6,7-dimethoxy-3-[({[4-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}piperazine-1-carboxylate
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propan-1-one
N-methyl-2-(morpholin-4-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
6-[1-(2-methyl-4-phenylpyridine-3-carbonyl)piperidin-3-yl]pyrimidin-4-ol
2-(3-methylpentanamido)-7-oxo-N-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-[2-(cyclooctylamino)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
(1R,5S)-6-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-{1-oxo-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-2-yl}-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
{2-oxo-2-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}urea
1-[4-(1H-imidazol-1-yl)benzoyl]-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
3,4,7-trimethyl-2-[4-(3-methylpyridin-4-yl)piperazine-1-carbonyl]-1H-indole
(1S,5R)-6-(cyclobutylmethyl)-3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(4-fluorophenoxy)-1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]pyrrolidin-2-one
1-{[2-(difluoromethoxy)phenyl]methyl}azepan-2-one
2-[(4-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)pyridine-3-carbonyl]morpholine
N-[2-(furan-2-ylmethoxy)phenyl]-8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
4-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-ethyl-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-1,3-oxazole-4-carboxamide
N-cyclopropyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
methyl 2-[8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-cyclohexyl-4-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]piperazin-2-one
ethyl[(1-methylpyrrolidin-3-yl)methyl](quinolin-2-ylmethyl)amine
(3aS,6aS)-2-(4-chlorobenzoyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-cyclohexyl-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
5-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-3-amine
1-(2-phenylphenyl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}urea
2-{1-cyclopentyl-4-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-({4-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
N-[2-(dimethylamino)ethyl]-5-methyl-N-[(3-methylthiophen-2-yl)methyl]pyridine-3-carboxamide
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]pyridin-3-ol
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-3-(pyrrolidin-1-yl)piperidine
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
5-methoxy-2-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-indole
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]propan-1-one