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2-(dimethylamino)-N-{2-oxo-4-[2-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
4-({[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-5-(hydroxymethyl)-2-methylpyridin-3-ol
3-[5-(2-hydroxyethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(morpholin-4-yl)propan-1-one
3-[5-(pyridin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-cyclopentyl-5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(1-{[5-chloro-3-methoxy-2-(propan-2-yloxy)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-ethylphenyl)urea
6-fluoro-3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinolin-4-ol
methyl 6-(naphthalen-1-ylmethyl)-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
(2S)-2-({1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazol-4-yl}formamido)-4-methylpentanamide
5-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]quinoxaline
2-{1-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]azetidin-3-yl}pyridine
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)acetamide
[1-(1-cyclobutanecarbonylpiperidin-4-yl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
7-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-2,7-diazaspiro[4.5]decane
1-[(4-methanesulfonylphenyl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
ethyl 3-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}butanoate
ethyl 2-[(3-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]carbamoyl}phenyl)amino]acetate
4-chloro-N,N-dimethyl-5-{[methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1,3-thiazol-2-amine
4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole
1-(3-acetylphenyl)-3-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}urea
2-{[4-methyl-1-(3-methylpyrazin-2-yl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
2-{1-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}ethan-1-ol
N-[2-(3-methoxyphenyl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-(1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)propanamide
2-benzyl-6-methyl-5-[5-(pyridazin-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
5-oxo-1-(pyridin-2-ylmethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxamide
(2R,3R,6R)-5-cyclopentyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3,5-dimethyl-1-({4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}methyl)-1H-pyrazole
2-methyl-5-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,3-thiazole
4-(hydroxymethyl)-1-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]piperidin-4-ol
4-(2-phenylethyl)-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({2-[5-(cyclohexylsulfanyl)furan-2-yl]-1H-imidazol-1-yl}methyl)-5-methyl-1,2,4-oxadiazole
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-(2-methoxyphenoxy)-N-methylacetamide
2-[4-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
1-ethyl-4-{[(7-methanesulfonyl-4-methylquinazolin-2-yl)(methyl)amino]methyl}pyrrolidin-2-one
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]ethan-1-one
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-(methoxymethyl)-N-[2-(N-methylmethanesulfonamido)ethyl]thiophene-2-carboxamide
(3S)-3-ethyl-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}morpholine
N-(2-methylpropyl)-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
N-[2-methyl-4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
(3R,4R)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
4-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
1-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-4-methyl-1,4-diazepan-5-one
(3S,4S)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-propylpyrrolidine-3-carboxylic acid