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N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]propan-1-one
(1R,5R)-3-methanesulfonyl-6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-benzyl-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-{[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-methylpyridine
4-({1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}methyl)morpholine
1,3,5-trimethyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-4-sulfonamide
(3aR,6aR)-2-methanesulfonyl-5-(naphthalene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 2-(diethylsulfamoyl)-6-(quinolin-4-ylmethyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1,6-dimethyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
1-[1-(propan-2-yl)piperidine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-[(2-fluorophenyl)methyl]-N-methyl-N-[4-(morpholin-4-yl)butyl]-1,3-benzoxazole-6-carboxamide
2-[1-(4-chlorophenyl)cyclopropyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]{[2-(methoxymethyl)pyrimidin-5-yl]methyl}amine
(2E)-3-(2,3-difluorophenyl)-1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)prop-2-en-1-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(9-methyl-9H-carbazol-3-yl)ethan-1-one
2-[(3-chlorophenyl)methyl]-4-{4-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-[1-(2-fluorophenyl)cyclopropanecarbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-{3,9-diazaspiro[5.5]undecan-3-yl}-4,4,4-trifluorobutan-1-one
N2-cyclobutyl-N4-(4-fluorophenyl)morpholine-2,4-dicarboxamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(2-methylphenyl)propan-1-one
4-{5-[(4-methylphenyl)sulfanyl]furan-2-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
methyl 4-{[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-benzyl-8-{[3-(furan-2-yl)phenyl]methyl}-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-chlorophenyl (7R,9aR)-7-[(4-hydroxyphenyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-(furan-2-yl)-2-{[1-(5-phenyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]amino}ethan-1-ol
3-hydroxy-3-({[1-(methoxymethyl)cyclopentyl]amino}methyl)-1-[(3-methoxyphenyl)methyl]piperidin-2-one
1-ethyl-4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
(3R,5S)-N3-(4-fluorophenyl)-N5-[(2-methoxyphenyl)methyl]-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
1-cyclopentyl-5-oxo-N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxamide
dimethyl(3-{2-[1-(quinoxalin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(thiophen-2-yl)azetidin-1-yl]ethan-1-one
methyl 2-[(4-fluorophenyl)sulfamoyl]-6-(3-phenylprop-2-ynoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
(4aS,7aR)-1-{[3-(cyclopentyloxy)phenyl]methyl}-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-4-(azepan-1-yl)-1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-3-ol
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
2-(dimethylamino)-N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-2-(4-fluorophenyl)acetamide
1-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]urea
(2S,4S)-4-[4-(4-chlorophenyl)butanamido]pyrrolidine-2-carboxylic acid
1'-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-ethyl-1H-pyrazole-4-carboxamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(pyrazin-2-yl)propanamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)oxane-4-carboxamide
1-(4-methyl-1H-imidazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
methyl (2R)-2-({2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxyphenyl}formamido)propanoate
1-[(2,3-difluorophenyl)methyl]-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine