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2-(furan-2-yl)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-1-methyl-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
2-ethyl-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
5-ethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1,3-oxazole-4-carboxamide
1-cyclopropanecarbonyl-N-(1-phenylpiperidin-4-yl)piperidine-4-carboxamide
8-(1,4-dithiepan-6-yl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
(3R,4S)-4-({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)amino)oxolan-3-ol
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
N-(3-chloro-4-propoxyphenyl)-4-(morpholin-4-yl)piperidine-1-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
ethyl 2-[({[2-(2-fluorophenoxy)pyridin-3-yl]methyl}carbamoyl)amino]acetate
N-[1-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-4-yl]methanesulfonamide
6-ethyl-N-[2-(ethylsulfanyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-benzyl-N3-cyclohexyl-N3-methyl-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2S,4R)-4-amino-1-(4-ethenylbenzoyl)-N-ethylpyrrolidine-2-carboxamide
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
5-{[benzyl(methyl)amino]methyl}-N-[(1-ethyl-1H-imidazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
(2-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}quinolin-3-yl)methanol
(4aS,8aR)-1-(2-aminoethyl)-N-[(2-fluorophenyl)methyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
3-(2-fluorophenyl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
1-cyclobutanecarbonyl-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
(4S)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
3-(3-fluorophenyl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]propan-1-one
8-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-methyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1-benzofuran-7-carboxamide
N-[(2,4-difluorophenyl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
methyl (2S,4R)-4-[2-(1H-indazol-1-yl)acetamido]-1-methylpyrrolidine-2-carboxylate
2-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-2,3-dihydro-1H-isoindole
2-(3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
3-({[(4-fluorophenyl)methyl](1-hydroxybutan-2-yl)amino}methyl)benzonitrile
4-[(2-hydroxyethyl)sulfanyl]-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]benzamide
ethyl 4-[(4,7-dimethyl-2-oxo-2H-chromen-6-yl)carbamoyl]piperazine-1-carboxylate
2-hydroxy-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(2,4,5-trimethoxyphenyl)methyl]amine
9-[3-(4-fluorophenyl)propanoyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]aniline
3-(1-butyl-1H-imidazol-2-yl)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidine
diethyl(3-{4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}propyl)amine
(3R,4R)-4-(azepan-1-yl)-1-(3-phenylpropyl)piperidin-3-ol
2-ethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
9-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
1-ethyl-4-{2-[3-(methoxymethyl)piperidine-1-carbonyl]-2,3-dihydro-1H-inden-2-yl}piperazine
1-[1'-(2-hydroxy-3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
9-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
2-(1H-indol-3-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-N-[(4-methoxyphenyl)methyl]propanamide
{5-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-2-propoxyphenyl}methanol