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N-cyclopropyl-4-{methyl[2-(pyridin-2-yl)ethyl]sulfamoyl}benzamide
2-(2-methoxyethyl)-4-{4-[2-(thiophen-3-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-[benzyl(methyl)amino]-3-{5-[(cyclohexylamino)methyl]-2-methoxyphenoxy}propan-2-ol
1-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-2-phenylethane-1,2-dione
6-{1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-2-amine
4-cyclopentyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]pyrimidin-2-amine
N1-[4-(propylsulfanyl)phenyl]piperidine-1,3-dicarboxamide
N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-yl}methyl)cyclopropanesulfonamide
(3S,4S)-4-(4-fluorophenyl)-1-(1H-indole-6-carbonyl)piperidin-3-ol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}ethan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)benzamide
N-(1H-indol-4-ylmethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
6-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)(1,3-thiazol-2-ylmethyl)amine
5-ethyl-2-{5-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
5-[4-(2-chlorophenyl)-2-methyl-5-oxopiperazine-1-carbonyl]pyridine-2-carbonitrile
ethyl 5-{[(1R,2R)-2-(benzyloxy)cyclopentyl]carbamoyl}-1H-imidazole-4-carboxylate
1-(cyclohexylmethyl)-4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
2-[(5-methylpyrazin-2-yl)methyl]-9-(6-methylpyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,5S)-N-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
ethyl 3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-4-(thiophene-2-carbonyl)piperazine
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
1-ethyl-4-[({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-methyl-3-({3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,2-oxazole
N-{[4-(aminomethyl)phenyl]methyl}-5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-amine
2-(dimethyl-1,2-oxazol-4-yl)-1-[2-(3-fluorophenyl)piperidin-1-yl]ethan-1-one
N-{[7-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
2-{1-[(2-methoxynaphthalen-1-yl)methyl]pyrrolidin-3-yl}acetic acid
N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(3R)-1-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}pyrrolidin-3-ol
[(2S,4R)-4-(dimethylamino)-1-[6-(propan-2-yl)-1H-indole-2-carbonyl]pyrrolidin-2-yl]methanol
4-(3-chloro-4-fluorophenyl)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole
2-[4-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperazin-1-yl]acetamide
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-ol
5-(3,4,5-trimethoxyphenyl)-1,2,3,4-tetrahydroisoquinoline
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-4-phenyl-1H-imidazol-5-yl}pyridine
methyl 4-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-4-oxobutanoate
2-(1,5-dimethyl-1H-pyrazol-4-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(2-chloro-4-fluorophenyl)methyl]-N-[(5-methylpyrazin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-(morpholin-4-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-4-amine
5-methoxy-2,4-dimethyl-N-[(1-methylpiperidin-3-yl)methyl]benzene-1-sulfonamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]-6-(4-fluorophenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
(4aR,7aS)-1-methanesulfonyl-4-[2-(pyridin-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole