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N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-4-(piperidin-3-ylmethyl)benzamide
N-[(3S,4R)-1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-(1H-1,3-benzodiazol-2-yl)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)propanamide
S-[4-(3-cyanopiperidine-1-carbonyl)phenyl]-3-hydroxypropane-1-sulfonamido
2-(pyridin-2-yl)-5-[5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyrimidine
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-6-methyl-N-(propan-2-yl)quinoline-4-carboxamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-(3-methoxypropyl)piperidine
1-(1-methyl-5-{[4-(morpholin-4-yl)piperidin-1-yl]methyl}-1H-pyrrol-3-yl)ethan-1-one
5-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-oxazole-4-carboxamide
(4aS,7aR)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-4-(pyridin-4-yl)pyrimidin-2-amine
5-{[2-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]methyl}-1-phenyl-1H-1,2,3,4-tetrazole
6-ethoxy-3-({methyl[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(4-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
1'-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1S,5R)-3-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-3,9-diazabicyclo[3.3.2]decan-10-one
N-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[4-(4-methoxy-2,3,6-trimethylbenzenesulfonamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
2-(3-hydroxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
(3S,9aR)-3-benzyl-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(5S,9aS,9bS)-5-(4-fluorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(1S,5R)-3-[(5-acetylthiophen-3-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]benzamide
5-({3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)-2-(3-methylphenyl)pyrimidine
N-(1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
N-methyl-1-(9H-purin-6-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
3-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-1-phenylurea
1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-3-[(dimethylamino)methyl]pyrrolidin-3-ol
(3S,4R)-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-(2-methoxyethyl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-6-oxopiperidine-3-carboxamide
2-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-3-[(pyridin-2-ylmethyl)amino]benzamide
4-{4-[3-(1H-pyrazol-1-yl)azetidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl}pyridine
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
N-[(3-hydroxypyrrolidin-3-yl)methyl]-3-methanesulfonylbenzamide
6-[3-(hydroxymethyl)pyrrolidin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-benzyl-9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-(diethylamino)-3-{2-methoxy-5-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
5-fluoro-2-{1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
1-[4-(ethanesulfonyl)piperazin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
5-benzyl-3-{[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
2-tert-butyl-6-[1-(methoxymethyl)cyclobutanecarbonyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(cyclohexylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[3-(3-methylphenyl)piperidin-1-yl]propan-1-one
5-(4-fluorophenyl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
6-[2-(4-fluorophenyl)piperidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-(3,4-difluorophenyl)-4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amine