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(1S,5R)-3-benzyl-6-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(2-methoxy-2-methylpropyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
8-[(5-cyclopentylthiophen-2-yl)methyl]-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,3R,6R)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
4-(2-amino-6-methoxypyrimidin-4-yl)-1-(3,5-dimethylphenyl)piperazin-2-one
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
[(1-ethylpyrrolidin-2-yl)methyl](furan-2-ylmethyl){[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
2-[(2-methoxyethyl)(methyl)amino]-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
5-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-N-propylpyrimidin-2-amine
8-[(2,3-difluoro-4-methylphenyl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
6-[(2-ethyl-1,3-thiazol-4-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
N-ethyl-4-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrimidine-5-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methanesulfonamidoacetamide
6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine-3-carbonitrile
4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-2-methoxyphenol
(3aR,5S,6S,7aS)-2-[2,2-dimethyl-1-(3-methylthiophen-2-yl)cyclopropanecarbonyl]-octahydro-1H-isoindole-5,6-diol
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-methyl-1,4-diazepan-5-one
4-(4-fluorophenoxy)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
N-({7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
1-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyrrolidin-2-one
9-methyl-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]-9H-carbazole-3-carboxamide
{4-[(4-methoxyphenyl)methyl]-1-(4-methoxypyrimidin-2-yl)piperidin-4-yl}methanol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-1-carboxamide
5-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylpiperidine-3-carboxamide
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
3-methyl-N-{3-[3-(1-methylpiperidin-3-yl)propanamido]phenyl}benzamide
5-chloro-4-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
N-methyl-N-[(5-methylfuran-2-yl)methyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,2-dimethyloxane-4-carboxamide
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-methyl-4-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]quinoline
3-cyclopropyl-1-methyl-5-[3-(trifluoromethyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
(3aS,6aS)-2-cyclopentyl-5-[2-(pyridin-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-carbamoylphenyl)-3-[(3-methylpiperidin-1-yl)methyl]benzamide
1-({2-[4-(morpholin-4-yl)butoxy]phenyl}methyl)azepan-4-amine
N-[(2,3-dimethoxyphenyl)methyl]-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
3-(2-fluorophenyl)-1-methyl-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1H-pyrazole
2-(cyclohex-1-ene-1-carbonyl)-1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-{[(3R,4R)-4-(hydroxymethyl)-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-yl]methyl}piperidin-4-ol
3-{[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]methyl}benzoic acid
1-[2-(2,3-dihydro-1H-inden-2-yl)acetyl]-1,4-diazepane-6-carboxylic acid
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine
(3S,4S)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-amino-4-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
1-[2-(quinolin-3-yl)pyrimidin-4-yl]piperidin-3-ol
2-amino-4-ethyl-N-[2-(N-methylmethanesulfonamido)ethyl]-1,3-thiazole-5-carboxamide
7-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2,7-diazaspiro[4.4]nonane-1,3-dione