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N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[3-(5-methylfuran-2-yl)-1H-indazol-1-yl]acetamide
2-{2-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methoxy]phenoxy}acetamide
5-(2-chlorophenyl)-N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}furan-2-carboxamide
1-{4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-(methylamino)ethan-1-one
(3R)-3-methyl-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
N-(2-methoxyethyl)-3-methyl-4-({[2-(2-oxoimidazolidin-1-yl)ethyl]carbamoyl}amino)benzamide
7-(2-benzyl-1,3-thiazole-4-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]-1-propylpiperidine
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
1-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)piperazine
3-{1-[(8-fluoroquinolin-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-2-[(2-fluorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
4-(2-methylquinolin-6-yl)-1-[(5-propylfuran-2-yl)methyl]piperidin-4-ol
2-[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]acetamide
5-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-N-methylthiophene-2-carboxamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-chloro-2-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
N,N-dimethyl-6-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazin-2-amine
N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
4-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-1-phenylpiperazin-2-one
(2S)-2-({1-[3-(4-fluorobenzenesulfonamido)phenyl]piperidin-4-yl}amino)-3-phenylpropanamide
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(3-phenylpropyl)benzamide
N-ethyl-3-methoxy-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)propanamide
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N,N-diethyl-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-benzyl-N3-cyclopropyl-N5-[2-(2-fluorophenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-2-(4-fluorophenyl)azetidine
N-[2-(4-ethylmorpholin-2-yl)ethyl]-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N,2,6,8-tetramethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(2-methoxyethyl)-2-(1-methylcyclohexanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
7-chloro-3-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cycloheptylacetamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(2-{2-[1-(2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-(2-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)acetamide
N-[1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
3-(4-fluorophenyl)-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
2-[methyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amino]-1-phenylethan-1-ol
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
7-(2,2-dimethylpropyl)-2-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-[2-(4-fluorophenoxy)ethyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
methyl 2-{8-[(4-hydroxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
methyl 4-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}-1H-pyrazole-3-carboxylate
2-(5-acetylthiophen-3-yl)-1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}ethan-1-one