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2-(5-chloro-2-methoxyphenyl)-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]acetic acid
N-methyl-5-phenyl-N-[1-(pyridin-2-yl)propan-2-yl]-1H-pyrrole-2-carboxamide
2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
(2S,4R)-4-amino-N-ethyl-1-{2-[(4-ethylcyclohexyl)formamido]acetyl}pyrrolidine-2-carboxamide
5-[4-(4-amino-6,7-dimethoxyquinazolin-2-yl)phenyl]imidazolidine-2,4-dione
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
1-[4-(2-phenylethyl)piperazin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
(1S,5R)-3-[(2-butyl-1H-imidazol-4-yl)methyl]-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
3-{2-[5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
3-[(3aS,6aS)-1-(2-fluorobenzoyl)-octahydropyrrolo[3,4-b]pyrrol-5-yl]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-(3-fluorophenoxymethyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
1-benzyl-4-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-6-methoxy-1,4-diazepan-2-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-(4-{[2-(3-phenylpropyl)morpholin-4-yl]methyl}thiophen-2-yl)ethan-1-one
1-[(3R,5R)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
3-{1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]azetidin-3-yl}pyridine
1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
ethyl N-[3-(4H-1,2,4-triazol-4-yl)phenyl]carbamate
3-({2-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-cyclopentyl-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-one
4-[4-(4-methylpiperazin-1-yl)benzoyl]-1,4-oxazepan-6-ol
1-(azepan-1-yl)-3-(4-chloro-2-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
3-[2-(2-methoxypyridin-3-yl)-4-methylphenyl]-1,3-oxazolidin-2-one
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-ethyl-1,3-dihydroxypropan-2-yl)-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-(4-chlorophenyl)-N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(oxolan-2-ylmethyl)cyclopropane-1-carboxamide
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-fluoro-N-(furan-2-ylmethyl)benzamide
1-{4-[2-cyclobutyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-methoxyethan-1-one
1-cyclopentanecarbonyl-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]piperidine-4-carboxamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
methyl 4-({4-[(1-methyl-1H-indol-3-yl)methyl]-7-oxo-1,4-diazepan-1-yl}methyl)benzoate
2-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-(1H-pyrrol-1-yl)propanamide
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)-1-methylpiperazin-2-one
N-[4-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenyl]acetamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}-6,8-dimethylquinolin-4-ol
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(2S)-1-hydroxybutan-2-yl]-1H-pyrazole-3-carboxamide
ethyl 1-(furan-3-carbonyl)-4-(2-phenylethyl)piperidine-4-carboxylate
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(pyridin-4-yl)quinoline-4-carboxamide
4-(1H-indol-5-yl)-N,N,5,6-tetramethylpyrimidin-2-amine
4-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-5,6,7,8-tetrahydroquinazolin-2-amine
1-[(1R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-4-(4-methyl-1,3-oxazole-5-carbonyl)piperazine
1-[(4-fluorophenyl)methyl]-N-[(4-phenyloxan-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide