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3-{[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
1-[ethyl(methyl)sulfamoyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
2-(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
2-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(1-benzyl-1H-imidazol-2-yl)-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidine
N-benzyl({4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}amino)sulfonamide
N-methyl-1-{[3-(naphthalen-2-yl)phenyl]methyl}pyrrolidine-3-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[1-(naphthalen-2-yl)ethyl]acetamide
N-[2-(diethylamino)ethyl]-N-ethyl-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-benzyl-N-methyl-3-(2-oxopyrrolidin-1-yl)piperidine-1-sulfonamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N6-cyclopropyl-N4-methyl-N4-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4,6-triamine
4-{[(4aS,7aR)-6,6-dioxo-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
2-({2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)benzonitrile
2-[methyl({[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
methyl 1-(2-methoxyethyl)-5-[(oxan-4-yl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(2H-1,3-benzodioxol-5-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenol
3-(1-hydroxypropan-2-yl)-5-methoxy-3,4-dihydroquinazolin-4-one
N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridazine-3-carboxamide
(3aR,6aS)-5-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
(4aR,7aS)-1-ethyl-4-{2-[3-(methylsulfanyl)phenyl]acetyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-3-[2-(thiophen-3-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3S)-1-[7-(furan-3-carbonyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
4-[(8-methoxy-2H-chromen-3-yl)methyl]-1-methylpiperazine-2-carboxylic acid
1-(4-fluorophenyl)-2,2-dimethyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]cyclopropane-1-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2-(6-chloropyridazin-3-yl)-8-methyl-2,8-diazaspiro[4.5]decane
2-(2-methoxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
3-[(2-methoxyethyl)(thiophen-2-ylmethyl)amino]propane-1,2-diol
3-methoxy-5-{[(5-methylpyrazin-2-yl)methyl]carbamoyl}benzoic acid
N-cyclopropyl-1-[1-(3-fluorobenzoyl)piperidin-4-yl]piperidine-3-carboxamide
N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1,3-thiazol-4-yl)ethyl]amine
4-methyl-2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-[1-ethyl-2-(2-fluorophenyl)-7-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]acetamide
(1S,5R)-6-(1H-indol-5-ylmethyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[1-(5-chloropyridine-3-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
(2R,3R,6R)-5-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[(pyridin-4-ylmethyl)sulfamoyl]-N-[(3R)-pyrrolidin-3-yl]benzamide
5-[(4-acetamidophenyl)methyl]-1-(2-hydroxyethyl)-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
4-cyclopropyl-6-(4-methoxy-4-phenylpiperidin-1-yl)pyrimidine
4-({1-[(4-fluorophenyl)methyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl}methyl)morpholine
N-[3-(cyclohexyloxy)propyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
(3S,5R)-1-[(3,4-dimethoxyphenyl)methyl]-N3-[3-(dimethylamino)propyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide