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1-(5-ethoxyfuran-2-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[5-(2-chloro-6-methoxyphenyl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
N-(3-{2-oxo-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethoxy}phenyl)propanamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-amine
1-(4-{4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)ethan-1-one
1-[2-(3-methoxypropyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(oxolan-3-yl)piperidine-4-carboxamide
3-fluoro-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-4-carboxamide
4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
4-{[(4aS,7aR)-4-(3-methylbut-2-en-1-yl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzoic acid
1-ethyl-4-{[methyl({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]methyl}pyrrolidin-2-one
6-methoxy-4-(thiomorpholine-4-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)piperidin-2-one
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
3-{5-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
4-(1-butyl-1H-imidazol-2-yl)-N-(4-fluorophenyl)piperidine-1-carboxamide
methyl 5-[4-({[(1R)-1-carbamoylethyl]amino}methyl)phenoxymethyl]furan-2-carboxylate
N-benzyl-2-(2-oxoazonan-1-yl)-N-(oxolan-2-ylmethyl)acetamide
4-(cyclohex-1-en-1-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
N-(1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-2-(1H-indol-3-yl)acetamide
3-{[cyclopropyl(6-methylpyridin-2-yl)methyl]carbamoyl}-5-methoxybenzoic acid
N-[1-(2-methanesulfonylethyl)piperidin-4-yl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
6-methoxy-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
2-(4-{[(furan-2-ylmethyl)(methyl)amino]methyl}phenyl)-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
3-{5-[(3,4-dimethoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-(pyridin-2-ylmethyl)urea
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-(1H-imidazol-1-ylmethyl)cyclopropane-1-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
9-(2,3-dihydro-1H-inden-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-3-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidine-1-carboxamide
N-cyclopropyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(quinoxaline-5-carbonyl)piperidine-3-carboxylate
9-[3-(ethylsulfanyl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-2,1,3-benzoxadiazole
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
3-(4-hydroxyphenyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-5-carboxamide
2-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-5-{4-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
5-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
1-ethyl-4-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-1H-indole
1-(3-propyl-1H-pyrazole-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
9-(4-fluorobenzoyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
3-(isoquinolin-5-yl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-ethyl-N-[3-(4-methoxyphenyl)propyl]-3,5-dimethyl-1H-pyrazole-4-carboxamide
5-methoxy-2-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
5-[(dimethylamino)methyl]-N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}furan-2-carboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[2-(thiophen-3-yl)acetyl]piperidine-4-carboxamide
1-{6-[({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridin-3-yl}ethan-1-one
2-(5-chloro-2-methoxyphenyl)-2-[(2-methoxyethyl)(methyl)amino]acetic acid