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1-[2-(dimethylamino)ethyl]-4-[4-(2-methylphenyl)piperazine-1-carbonyl]pyrrolidin-2-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-(4-methylphenyl)propan-1-ol
2-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-{2-oxo-2-[3-(3-phenylpropanoyl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
5-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
N-(4-butanamido-3-methoxyphenyl)-2-oxo-2H-chromene-3-carboxamide
2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-N-(propan-2-yl)propanamide
(4aS,8aR)-6-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-(4-ethyl-1H-pyrazol-5-yl)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
methyl 2-[(butan-2-yl)sulfamoyl]-6-[(4-hydroxy-3,5-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-ethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-[2-(2-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1H-imidazol-1-yl)ethyl]pyridine
2-(2-{[2-(oxan-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-methoxy-5-sulfamoylbenzamide
1-(oxolane-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-butyl-2-[(5-ethylpyrimidin-2-yl)(methyl)amino]acetamide
6-tert-butyl-2-{2-[(2-methylpyrrolidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-3-yl)ethan-1-one
2-(2-ethoxyphenyl)-1-(prop-2-en-1-yl)-1H-imidazole
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(thiophen-3-ylmethyl)-1,2-oxazole-3-carboxamide
ethyl 2-(1-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-2-yl)acetate
1-[(4aR,8aS)-1-[2-(2-chloro-4-fluorophenyl)acetyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
9-methyl-3-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-3,9-diazaspiro[5.6]dodecane
2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(pyrrolidine-1-sulfonyl)-decahydro-1,6-naphthyridin-2-one
(1S,5R)-6-benzyl-3-(2-methoxypyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(1H-indazol-1-yl)ethan-1-one
1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
methyl 1-[(3S,5S)-5-{[(4-methoxyphenyl)methyl]carbamoyl}-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-methyl-6-(piperidin-4-yl)-N-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]pyrimidin-4-amine
2-{1-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperidin-2-yl}acetamide
N-cyclopropyl-N-{[7-fluoro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-3-(2-methoxyphenyl)propanamide
N-{1-[1-(furan-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
1,6-dimethyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-(4-phenyl-1,3-thiazol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(4-methyl-1H-pyrazol-1-yl)propanamide
6-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(pyridin-2-yl)propanamide
3-(cyclopropylmethyl)-1-(3-fluoropyridin-2-yl)piperidine-3-carboxylic acid
9-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-6-oxa-9-azaspiro[4.5]decane
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
2-[3-(benzyloxy)propyl]benzene-1-sulfonamide
[7-fluoro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[4-methyl-2-({[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amino)pyrimidin-5-yl]ethan-1-one
9-[(2S)-2-amino-3-hydroxypropanoyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one