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3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[2-(2-phenylethyl)piperidin-1-yl]propan-1-one
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
1-({5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]furan-2-yl}methyl)-1H-pyrazole
5-(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-[(4-fluorophenyl)methyl]-4-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)butanamide
N-{2-[2-(trifluoromethoxy)phenyl]ethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-phenyl-5-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-benzyl-6-methyl-2-oxo-N-(1,3-thiazol-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
(3S)-1-[1-methyl-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}furan-2-carboxamide
3-({[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
4-[(2-chlorophenyl)methyl]-11-[(2-hydroxyethyl)(methyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{4-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)methyl]thiophen-2-yl}ethan-1-one
N,N-diethyl-1-[(1s,4s)-4-[3-(3,4-dimethoxyphenyl)propanamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(5-chloro-1H-indol-2-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-(azocan-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)acetamide
3-(4-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)phenol
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]-2,1-benzoxazole-3-carboxamide
methyl({2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl})(2-phenylethyl)amine
1-(furan-2-ylmethyl)-4-[4-(3-methoxyphenyl)-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl]piperidine
5-[({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
2-({2-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]phenyl}amino)acetic acid
(4aS,8aR)-6-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(2-methyloxolan-2-yl)methyl]propanamide
(3S,4R)-1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
6-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
3,5-dimethyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-1,2-oxazole-4-sulfonamide
2-[4-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidin-1-yl]acetamide
7-(1-benzothiophen-2-ylmethyl)-3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-(2H-1,3-benzodioxol-4-ylmethyl)-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(2-ethyl-1H-imidazol-1-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-{4-[benzyl(2-hydroxyethyl)amino]piperidin-1-yl}-N-(1-phenylethyl)benzamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-decahydro-1,6-naphthyridin-2-one
N-{2-[(2-methyl-1H-imidazol-1-yl)methyl]phenyl}-2-(morpholin-3-yl)acetamide
4-{1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}quinoline
2-{[2-(2-phenylethyl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
4-ethyl-1-methyl-3-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[(2-methyl-1-benzothiophen-3-yl)methyl]azetidin-3-yl}morpholine
2-{1-[(4-fluorophenyl)methyl]-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]({2-phenylimidazo[1,2-a]pyridin-3-yl}methyl)amine
1-(carbamoylmethyl)-N-{3-[(4-chlorophenyl)sulfanyl]propyl}piperidine-3-carboxamide
6-[4-(1H-imidazol-2-yl)piperidin-1-yl]-9H-purine
2-methoxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-3-carboxamide
1-{3-[3-(2-phenylethyl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
3-{[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)piperidin-4-yl]oxy}pyridine
2-{[(1-methyl-4-phenylpiperidin-4-yl)methyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-cyclopropyl-N-(3-fluorophenyl)-1H-1,2,4-triazole-5-carboxamide
4-(4-phenyl-1H-imidazol-5-yl)-2,1,3-benzothiadiazole