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2-(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
4-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]morpholine
methyl 6-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-(2-ethyl-6-methylphenyl)pyrrolidin-2-one
N-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)-3-acetamidopyrrolidine-1-carboxamide
(2-{2-[1-(7,8-dimethylquinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-5,6,7,8-tetrahydroquinoline-3-carboxamide
6-{[4-(dimethylamino)azepan-1-yl]sulfonyl}-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
N-{4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]phenyl}-N-methylmethanesulfonamide
6-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-N-ethyl-N-methylpyridine-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[5-(azepan-4-yl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N,N-dimethylpropanamide
(1S,5R)-1,3,3-trimethyl-6-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
(1S,5R)-3-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]cyclobutanecarboxamide
7-[cyclohexyl(methoxy)methyl]-4-[2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-methoxy-4-(propan-2-yloxy)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[4-(pyrrolidine-1-carbonyl)phenoxy]-1-(thian-4-yl)piperidine
N-[5-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)carbamoyl}amino)-2-fluorophenyl]-2-methylpropanamide
(3aR,6aS)-5-(2-fluoro-6-hydroxybenzoyl)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
1-(2-methylphenyl)-4-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}piperazine
(3S,4S)-4-cyclopropyl-1-[4-(4-methoxyphenyl)-4-oxobutanoyl]pyrrolidine-3-carboxylic acid
N-cycloheptyl-3-[methyl(2-methylprop-2-en-1-yl)amino]propanamide
4-hydroxy-2-(4-methylphenyl)-N-[3-(oxolan-3-yl)propyl]pyrimidine-5-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-[4-(3-methylpiperidine-1-carbonyl)phenyl]urea
2,4-dimethyl-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-1,3-oxazole-5-carboxamide
4-{1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-phenyl-1,3-oxazole
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-N-(2-methylpropyl)-5-[(pyridin-3-yloxy)methyl]piperidine-3-carboxamide
4-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-1-phenylpiperazin-2-one
2,6-dimethyl-3-[4-(pyrazin-2-yl)piperazine-1-carbonyl]quinoline
ethyl 4-({2-[4-(methoxycarbonyl)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)piperazine-1-carboxylate
2-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-4-(propan-2-yl)-1,3-thiazole
4-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-6-(4-methyl-1H-pyrazol-1-yl)pyrimidine
6-({1-[ethyl(methyl)amino]cyclohexyl}methyl)-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
4-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
2-[1-(3-methylbut-2-en-1-yl)-4-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperazin-2-yl]ethan-1-ol
(2H-1,3-benzodioxol-4-ylmethyl)[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amine
N-(2-aminoethyl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
1-(2-{1-[(2R)-2-amino-2-phenylacetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(oxolane-3-carbonyl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
N-[2-(dimethylsulfamoyl)ethyl]-2-(methylamino)pyridine-4-carboxamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[2-(1H-pyrazol-4-yl)ethyl]piperidine
4-hydroxy-2-(4-methylphenyl)-N-(oxan-3-yl)pyrimidine-5-carboxamide
6-ethyl-N2,N2,N4-trimethyl-N4-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrimidine-2,4-diamine
N-ethyl-N-(2-methylprop-2-en-1-yl)-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
4-[3-(5-methylfuran-2-yl)-1-phenyl-1H-pyrazol-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one