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{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(2-methoxyethyl)methylamine
N-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-5-[1-(oxane-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-{1-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]piperidin-4-yl}pyrrolidin-2-one
2-butyl-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
2-[(3,5-difluorophenyl)methyl]-8-(2-propoxyethyl)-2,8-diazaspiro[4.5]decan-3-one
1-(cyclopropylmethyl)-5-(2,3-dimethoxybenzoyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)-3-(2-oxopiperidin-3-yl)urea
N-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-4-(piperidin-3-yl)benzamide
2-(2-chloro-4-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}phenoxy)acetamide
(3S,4R)-4-(4-fluorophenyl)-1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
2-[5-(3-methylthiophene-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-1,3-benzodiazole
(1S,5R)-3-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[1-(4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-2-yl]ethan-1-ol
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
1-(2-fluorobenzenesulfonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-(morpholin-2-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-methyl-4-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholine-4-carbonyl)pyridin-2-amine
(2S)-2-{4-[2-methoxy-5-(propan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}-3-methylbutanamide
4-(4-fluorophenyl)-1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidin-4-ol
3-(3-hydroxy-3-methylbutyl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
8-(5-methoxyfuran-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl})amine
(1r,4r)-4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)cyclohexan-1-ol
2-ethoxy-5-{2-[3-(methylcarbamoyl)pyrrolidin-1-yl]pyrimidin-4-yl}benzoic acid
2-(cyclopropylmethyl)-8-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-2-hydroxybenzoic acid
5-({[(3-{2-[4-(2,3-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
1-ethyl-N-[3-(2-ethylphenoxy)propyl]-N-methyl-1H-pyrazole-5-carboxamide
methyl (2S)-3-methyl-2-({5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazol-3-yl}formamido)butanoate
2-{1-[(2-fluorophenyl)methyl]-4-(quinolin-2-ylmethyl)piperazin-2-yl}ethan-1-ol
2-amino-4-(1-ethyl-1H-indol-6-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(2-methylphenyl)pyrrolidin-3-ol
3-methoxy-1-[2-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}amine
N-[(5-methoxy-1H-indol-2-yl)methyl]-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3,5-dichloro-4-{[2-(methoxymethyl)piperidin-1-yl]methyl}pyridine
1-[1-(furan-3-ylmethyl)pyrrolidin-3-yl]-4-methylpiperazine
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-5-methyl-1,3-benzoxazole
1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-5-phenyl-1H-pyrrole-2-carboxamide
5-[3-(1H-indol-3-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
5-cyclobutyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1,3,4-oxadiazol-2-amine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-[(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]pyridine
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-(propan-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(2,3-dimethylphenyl)-3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3-oxopropanamide
2-chloro-4-{1-[3-(morpholin-4-yl)propyl]-1H-imidazol-2-yl}phenol
1-(azocan-1-yl)-3-[5-({[(3-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,6-dimethyl-2-(pyridin-3-yl)pyrimidin-4-amine
2-[1-(5-propylpyrimidin-4-yl)pyrrolidin-3-yl]benzoic acid
3-[({1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidin-4-yl}oxy)methyl]pyridine