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1-(2-oxo-2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-1,2-dihydropyridin-2-one
1-(4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(1H-pyrazole-3-carbonyl)-1,4-diazepane
2-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2,4-difluoro-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methoxybenzamide
1-(2-methoxyethyl)-2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-imidazole
N-{[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
2,3,5-trimethyl-N-[(6-methylquinolin-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
(3aR,6aR)-2-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclohexyl-9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(morpholin-4-yl)ethan-1-one
2-(2-chloro-6-methoxyphenyl)-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
1-(4-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
3-(1,4-diazepane-1-carbonyl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}benzene-1-sulfonamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
5-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
6-[(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)amino]-N,N-dimethylpyridine-3-carboxamide
2-{4-[2-(benzyloxy)acetyl]morpholin-3-yl}-N-(oxan-4-yl)acetamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-[4-(propan-2-yloxy)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
4-(2-methyl-1H-imidazol-1-yl)-1-(morpholine-4-sulfonyl)piperidine-4-carboxylic acid
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-pyrazole-4-carboxamide
1-(3-{[(8-chloro-4-hydroxyquinolin-2-yl)methyl]amino}propyl)pyrrolidin-2-one
4-(benzyloxy)-1-[4-(pyrazin-2-yl)piperazin-1-yl]butan-1-one
4-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-{[4-(dimethylamino)oxan-4-yl]methyl}-3-(2-phenylphenyl)urea
4-(2-{5-[4-(prop-2-en-1-yloxy)phenyl]-2H-1,2,3,4-tetrazol-2-yl}acetyl)-1,4-diazepan-2-one
N-(1-methyl-1H-pyrazol-4-yl)-2-[(1-methylpiperidin-4-yl)(2-phenylethyl)amino]acetamide
N2-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrimidine-2,4-diamine
6-[(diethylamino)methyl]-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(4-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}phenyl)methanol
N,2-dicyclopropyl-N-[(3-methoxyphenyl)methyl]pyrimidine-5-carboxamide
5-methyl-2-(5-methylthiophen-2-yl)-4-[(2-propyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-(2-chlorophenyl)-2-hydroxy-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
2-{5-[(1,4-dimethylpiperazin-2-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-methyl-5-{3-oxo-3-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propyl}pyrrolidin-2-one
3-[3-(4-phenylbenzoyl)piperidin-1-yl]propanamide
(1R,7S)-6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-3-(2-methoxyethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(thiophen-2-yl)propanamide
1-(2-chlorophenyl)-5-methyl-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
2-(4-acetylphenoxy)-1-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}ethan-1-one
6-methoxy-3-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl][(5-methyl-1H-1,2,4-triazol-3-yl)methyl]amine
(1R,5R)-6-(2-methoxyethyl)-3-(2-phenoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2-chloro-6-fluorophenyl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-4-methoxy-2-methylbenzamide
N-{3-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]phenyl}acetamide
2-(4-chloro-1H-indazol-1-yl)-6-fluorobenzamide
2-[5-({[(2-chlorophenyl)methyl]sulfanyl}methyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-3-yl]acetamide