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N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(3-phenylpropyl)piperidin-4-yl]propanamide
(3S,4R)-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[4-(2,3-dihydro-1-benzofuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-phenylpropan-1-ol
8-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[4-(2-methoxyphenyl)piperidin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-[(2S)-1-methoxypropan-2-yl]-3-[methyl(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-methoxy-3-methyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1-benzofuran-2-carboxamide
N-cyclopropyl-2-[4-({[2-(4-methyl-1,3-thiazol-2-yl)ethyl]carbamoyl}amino)phenyl]acetamide
3-{5-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-(2-hydroxyethyl)propanamide
7-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-(2-{6-azaspiro[2.5]octan-1-ylformamido}ethyl)-4-fluorobenzamide
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-{[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}acetamide
ethyl 2-{1-methyl-9-pentanoyl-1,4,9-triazaspiro[5.5]undecan-4-yl}acetate
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
2-[4-(2-methylquinolin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
8-(7-chloro-2-methylquinoline-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(pyrimidin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-N-[1-(naphthalen-1-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(2-{[methyl(oxan-4-yl)amino]methyl}phenoxy)ethan-1-ol
N-ethyl-2,3,4-trimethoxy-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
4-({4-methyl-5-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-[4-({4-[4-(methylamino)pyrimidin-2-yl]piperazin-1-yl}methyl)phenyl]prop-2-yn-1-ol
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
2-(1-ethylpiperidin-4-yl)-N-{2-[4-(trifluoromethyl)phenyl]ethyl}acetamide
2-ethyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)pyrimidine-5-carboxamide
N,N-diethyl-1-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
2-[4-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
1-(2-ethoxyethyl)-N-methyl-N-(2-methylpropyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(butylsulfanyl)-6-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]pyrimidin-4-amine
(3S)-N,N-dimethyl-1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]azepan-3-amine
7-(1,3-benzothiazol-2-yl)-4-[(2R)-oxolane-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-benzyl-5-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}pyrimidin-2-amine
(1S,5R)-6-benzyl-3-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-N-methyl-1-(oxan-4-yl)-4-{pyrazolo[1,5-a]pyridine-3-amido}pyrrolidine-2-carboxamide
2-phenyl-1-[1-(quinoline-4-carbonyl)piperidin-4-yl]ethan-1-ol
5-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-1,2-dihydropyridin-2-one
1-(cyclohexylmethyl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
1-[5-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N3-cyclohexyl-1-cyclopropyl-4-oxo-N5-[phenyl(pyridin-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-(pyrrolidin-3-yl)pyridin-2-amine
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetic acid
(3R,4S)-4-(4-methoxyphenyl)-1-[2-(methylsulfanyl)benzoyl]pyrrolidin-3-amine