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1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
1-(4-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
(2S,4S)-4-[(adamantan-2-yl)amino]-1-[(3-chlorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
1-{2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}azetidin-3-ol
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-(2,3,6-trimethylphenoxy)acetamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
3-({[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
2-(3-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}phenoxy)acetamide
2-(2-aminopyrimidin-5-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
2-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)thiophene-3-sulfonamide
2-(3-fluorophenoxy)-1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]piperidine-1-carboxamide
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-4-(1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)benzamide
8-[2-(3-acetyl-1H-indol-1-yl)acetyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-phenoxypropanamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methoxy-3-methylbenzoyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
6-ethyl-2-methyl-N-[3-(oxolan-3-yl)propyl]quinoline-4-carboxamide
1-methanesulfonyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
benzyl (1S,5R)-6-[(dimethylcarbamoyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxylate
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(1R,2S)-2-phenylcyclopropyl]-1,2-oxazole-3-carboxamide
3-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
N-ethyl-N-(oxan-2-ylmethyl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
2-[(2-ethylpyrimidin-5-yl)methyl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-{[4-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-{[4-(dimethylamino)-1-ethylpiperidin-4-yl]methyl}-4-methylpyrimidin-2-amine
butyl 4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxylate
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(2-chloro-6-methylphenoxy)ethyl]acetamide
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-1,2-oxazole-5-carboxamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N,2,8-trimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]quinoline-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
[2-(2-ethylphenyl)pyridin-4-yl]methanol
1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperidine-3-carbonitrile
4-(2-ethoxypyridin-3-yl)-6-(morpholin-4-yl)pyrimidin-2-amine
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine
4-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperazine-1-sulfonamide
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-methyl-2-phenylpyrimidine-5-carboxamide
ethyl 4-(5-propyl-1,2-oxazole-3-carbonyl)piperazine-1-carboxylate
5-ethyl-2-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]pyrimidine
5-chloro-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}pyridine-2-carboxamide
6-{3-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
ethyl 4-[(3-fluorophenyl)methyl]-1-(1,3-thiazole-4-carbonyl)piperidine-4-carboxylate
5-ethanesulfonamido-N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-1-methyl-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
({2-[4-(1H-imidazol-1-yl)butoxy]phenyl}methyl)dimethylamine