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(4aR,7aS)-1-ethyl-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
3-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]sulfonyl}pyridine
(1R,5R)-6-[(2,3-dimethoxyphenyl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-{2-[2-(prop-2-en-1-yl)phenoxy]ethyl}oxolane-3-carboxamide
N-methyl-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1-{3-[({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}amino)methyl]phenyl}ethan-1-one
(3S,4R)-1-(3-chloro-4-fluorobenzoyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-{1-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,3-triazol-1-yl]ethyl}-3-(2-methylpropyl)-1,2,4-oxadiazole
1-[2-(4-chlorophenyl)ethyl]-5-(4-methylpiperazine-1-carbonyl)piperidin-2-one
4-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-3-methoxybenzamide
(1S,4S)-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
4-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-5-methylpyrimidine
2-{2-[(4-phenylbutan-2-yl)amino]ethyl}-1,2-dihydrophthalazin-1-one
{9-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(furan-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
2-{2-[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidine
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
1-[2-(2-fluorophenoxy)phenyl]-3-[2-(morpholin-4-yl)butyl]urea
(3S,9aR)-8-(2-chlorobenzoyl)-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(methoxymethyl)-N,5-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
2-[4-(3-methyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
N,N-dimethyl-7-(1,3,7-trimethyl-1H-indole-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}phenoxy)propan-2-ol
2-chloro-4-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-6-methoxyphenol
1-cyclopentyl-4-({3-methyl-1-[2-(4-methylpiperazin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)piperazine
(3S,5S)-1-[(2,4-difluorophenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
{1-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
5-({[3-(4-fluorophenyl)oxolan-3-yl]methyl}amino)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{[4-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-3-amine
1-(carbamoylmethyl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-4-carboxamide
(2S)-2-{[(8-chloro-4-hydroxyquinolin-2-yl)methyl]amino}-2-phenylacetamide
1-(furan-2-ylmethyl)-3-[4-(naphthalen-1-yl)-1H-pyrazol-5-yl]piperidine
5-(4,4-difluoropiperidine-1-carbonyl)-2-ethylpyrimidine
methyl 4-(5-methyl-4-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}-1,3-oxazol-2-yl)benzoate
4-(2-methoxyphenoxy)-1-[3-(methylcarbamoyl)pyridin-2-yl]piperidine-4-carboxylic acid
(1S,5R)-6-methyl-3-(2-methylpyridin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(2-hydroxy-5-methylbenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2R,5R)-2,5-dimethyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine
N-(1-{7-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)oxolane-3-carboxamide
2-(4-{[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-yl)pyrimidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylbenzamide
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(methylamino)acetamide
(9aS)-2-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
ethyl 1-[2-(1H-indazol-1-yl)acetyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
1-{6-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
(4aS,8aR)-1-(3-hydroxypropyl)-6-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-decahydro-1,6-naphthyridin-2-one