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N-[2-(1,3-thiazol-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methyl-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
4-cyclopentanecarbonyl-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-{2-[(6,7-dimethoxy-4-methylquinolin-2-yl)amino]ethyl}methanesulfonamide
(2,1,3-benzothiadiazol-5-ylmethyl)({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
6-ethyl-2-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}quinoline-4-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carboxamide
2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-4-(pyridin-2-yl)pyrimidine
2-(4-fluorophenyl)-4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]morpholine
4-(difluoromethoxy)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]benzamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-cyclopropyl-N-({5,8-dimethoxy-2-[methyl(thiophen-2-ylmethyl)amino]quinolin-3-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
2-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}-N,N-dimethylbenzamide
11-{[3-(1H-imidazol-1-yl)propyl]amino}-4-[(4-methylphenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3S,9aR)-8-[(4-chlorophenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[(4-benzylpiperidin-1-yl)methyl]-2-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
N-({5-[(3-chloro-4-ethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-methylacetamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-hydroxy-N-methyl-4-oxo-4H-pyran-2-carboxamide
(1R,2R,4R)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
methyl 5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1-methyl-1H-pyrazole-3-carboxylate
N'-(5-chloro-2-methylphenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}propanediamide
[(5-chloro-2-ethoxyphenyl)methyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N,6-diethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
methyl(oxolan-3-ylmethyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
ethyl 1-[1-(4-hydroxyphenyl)propan-2-yl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-{2-[(3-methoxyphenyl)methyl]morpholin-4-yl}-4-phenylbutane-1,4-dione
3-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indazole
1,3-dimethyl-N-[1-(pyrazin-2-yl)propan-2-yl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(4aS,8aR)-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
8-(1,3-benzothiazol-2-ylmethyl)-3-benzyl-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,6-dihydroxy-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]benzamide
N-[2-(ethanesulfonyl)ethyl]-2,3-dimethyl-1H-indole-5-carboxamide
1-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(2-methoxyphenyl)propan-1-one
3-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-1-(3-fluoro-4-methylphenyl)urea
4-[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]-N-[2-(methylsulfanyl)phenyl]-4-oxobutanamide
N-(3-phenoxypropyl)-1-(propan-2-yl)piperidin-4-amine
(1S,5R)-3-[(2E)-but-2-en-1-yl]-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4S)-1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(naphthalen-2-yl)piperidin-3-ol
3-(cyclobutylsulfamoyl)-N-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]benzamide
3-{[6-(aminomethyl)-2-methylpyrimidin-4-yl](methyl)amino}-1-phenylpropan-1-ol
2-(3-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-amine
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
(2S,4R)-4-hydroxy-1-{[2-(propan-2-yloxy)naphthalen-1-yl]methyl}pyrrolidine-2-carboxylic acid
5-(3-chloropyridin-2-yl)pyridin-3-amine
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-3-chloro-4-methoxybenzamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylsulfanyl)ethan-1-one