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(1S,5R)-6-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-5-[(4-fluorophenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
N-{[1-(3-cyclopentylpropyl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
4-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}morpholine
4-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)benzoic acid
2-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-4-methoxyphenol
1-{3-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-4-(2-oxopyrrolidin-1-yl)butanamide
3-{4-[(5-acetylthiophen-3-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
N,1-dimethyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
6-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-1,4-oxazepan-6-ol
2-[3-({[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}amino)phenyl]-N-methylacetamide
{imidazo[1,2-a]pyridin-2-ylmethyl}(4-methoxy-4-methylpentan-2-yl)amine
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(pyridin-4-ylmethyl)(thiophen-3-ylmethyl)amine
2-{[5-(1-methoxyethyl)-4-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-{1-[(3-chlorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}-N-cyclopentylpropanamide
2-(4-{4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanoyl}morpholin-3-yl)acetic acid
methyl 2-[3-oxo-4-(prop-2-en-1-yl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetate
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(pyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1H-imidazol-1-ylmethyl)-1-[2-(phenylamino)pyrimidine-5-carbonyl]piperidin-4-ol
1-methyl-5-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)piperidin-2-one
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-methyl-1H-indol-1-yl)propan-1-one
1,3-dimethyl-6-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(5-methylfuran-2-yl)methyl]-2-(pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}-1,4-oxazepane
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(morpholin-4-yl)ethyl]amino}methyl)piperidin-2-one
1-(1H-imidazol-4-ylmethyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-(2-ethoxypyridin-3-yl)pyridine-3-carboxamide
1-(adamantane-1-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
3-hydroxy-1-(2-methoxyethyl)-3-[(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]piperidin-2-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-methoxypyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(4-methoxyphenyl)phenyl]-1-(oxane-4-carbonyl)pyrrolidine-2-carboxamide
6-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
N-{[(2S,4S)-4-fluoro-1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)pyrrolidin-2-yl]methyl}-3,3-dimethylbutanamide
4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methylphenol
N-{2-[(1-ethyl-5-oxopyrrolidin-3-yl)formamido]ethyl}-4-fluorobenzamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-(4-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}phenyl)acetamide
2-(2-amino-4-methyl-1,3-thiazol-5-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
(3R,4S)-4-cyclopropyl-1-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]pyrrolidin-3-amine
2-amino-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-6-(1H-indol-3-yl)pyridine-3-carbonitrile
6-({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
1-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-3-(2-methylphenyl)pyrrolidin-3-ol
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
3,4,5-trimethoxy-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
1-[2-(1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
3-(1,3-benzothiazol-2-yl)-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol