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1-[5-(cyclopropylmethyl)-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-3-ol
N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indazole-3-carboxamide
4-amino-N-(2-phenylphenyl)azepane-1-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-1,3-oxazole-5-carboxamide
(3R,5S)-N-butyl-1-[(3,4-dimethoxyphenyl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]piperidine-3-carboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidine
3-{[(cyclopropylmethyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
6-methyl-5-[5-(oxolan-3-yl)-1,2,4-oxadiazol-3-yl]-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methoxy-2-methylpropanamide
N-[(3S)-2-oxoazepan-3-yl]-5-phenoxyfuran-2-carboxamide
2-amino-N,6-dimethyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidine-4-carboxamide
N-(furan-2-ylmethyl)-2-(2-oxo-1,3-oxazolidin-3-yl)-N-(2-phenylethyl)acetamide
1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-propoxypiperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentyl-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
dimethyl({3-[2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]propyl})amine
N-ethyl-2-methyl-6-(piperidin-3-yl)-N-(pyridin-4-ylmethyl)pyrimidin-4-amine
1-(2-ethoxyethyl)-3-[(4-fluorophenyl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
2-methoxy-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-5-sulfamoylbenzamide
N-[3-(cyclopentyloxy)propyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-{5-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
methyl 6-benzyl-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
7-(5-fluoropyrimidin-2-yl)-4-(1,2,3,6-tetrahydropyridin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
(2S)-N-(2-methyl-1,3-benzothiazol-6-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
2-[3-(isoquinolin-5-yl)-4-methoxyphenyl]ethan-1-amine
3-({1-[1-(hydroxymethyl)cyclopropanecarbonyl]pyrrolidin-3-yl}methyl)benzamide
3-ethyl-4-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-pyrazole-5-carboxamide
methyl 3-chloro-4-({[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)carbamoyl}amino)benzoate
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]acetamide
1-[4-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
2-(4-{[4-(9-methyl-9H-carbazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
N-[(3-fluorophenyl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(pyrazin-2-yl)piperidin-3-amine
4-{[1-(2-propoxybenzoyl)piperidin-4-yl]methyl}morpholine
(2S,3R)-3-hydroxy-2-{4-[4-methoxy-3-(prop-2-en-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}butanoic acid
4-butyl-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)benzonitrile
4-propyl-5-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrimidine
1-methyl-4-[5-(piperidin-1-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]-1,4-diazepane
N-ethyl-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
1-[cyclohexyl(methyl)amino]-3-[3-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[2-(4-ethylmorpholin-2-yl)ethyl]-3-(2-methoxy-5-methylphenyl)urea
N-[2-(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)ethyl]acetamide
N3-[(1R)-1-(3-methoxyphenyl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[3-(morpholin-4-yl)propyl]acetamide
4-(4-ethoxy-3-methylphenyl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}butanamide
2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]quinoline
3-(2-methoxyphenyl)-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-5-carboxamide