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N-[5-(cyclopropylcarbamoyl)-2-methoxyphenyl]-4,4-difluoropiperidine-1-carboxamide
N-{[5-chloro-2-(propan-2-yloxy)phenyl]methyl}-4-(2-oxopyrrolidin-1-yl)butanamide
2-[2-(phenylamino)pyrimidine-5-carbonyl]-1,2-oxazolidin-4-ol
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-cyclopropyl-5-[2-(1H-pyrrol-1-yl)ethyl]-1H-1,2,4-triazole
4-(4-chlorophenyl)-1-[6-(methoxymethyl)pyridine-2-carbonyl]piperidin-4-ol
2-(4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-2-oxopiperazin-1-yl)benzonitrile
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-(phenylsulfanyl)ethan-1-one
2-(3-fluorophenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(dimethylamino)-4-methyl-N-[3-(pyridin-3-yloxy)propyl]pyrimidine-5-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
1-{2-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
1-(2-chloro-5-methylbenzoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-(methylsulfanyl)benzamide
2-(dimethylamino)-2-(4-methylphenyl)-1-{3-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
2-(2-amino-9H-purin-6-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-{1-[3-(dimethylamino)propanoyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-methyl-7-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
{[(3S,4R)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-(2,4-difluorophenyl)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-oxazole
1-methyl-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
3-[(2-methoxyethyl)sulfamoyl]-5-[3-(thiophen-2-yl)-1H-pyrazol-1-yl]benzoic acid
1-[1-(furan-3-ylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-[1-(1H-1,3-benzodiazol-2-yl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
2-(1,3-thiazolidine-3-carbonyl)-3,4-dihydroquinazolin-4-one
1-(furan-3-carbonyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(1,4-oxazepan-4-yl)butan-1-one
2-benzyl-9-[2-hydroxy-4-(methylsulfanyl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-4-{[(3-chlorophenyl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
{2-[4-(1,3-benzothiazol-2-yl)morpholin-2-yl]ethyl}dimethylamine
2-[1-(morpholin-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-1H-indole
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-(9H-purin-6-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)piperidin-4-amine
5-[3-(4-fluorophenyl)phenyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
[3-(2-methoxyethyl)-1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl]methanol
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-3-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
6-[(diethylamino)methyl]-N-methyl-N-[1-(pyridin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
N-[(5-chloro-2-methoxyphenyl)methyl]-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
2-(4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl)acetic acid
6-methyl-2-[(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)amino]-3,4-dihydropyrimidin-4-one
N-(cyclohex-1-en-1-ylmethyl)-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
1-(3-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenyl)ethan-1-one
N,N,2-trimethyl-7-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(4-fluorophenyl)pyridine-3-carboxamide
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[(3-fluorophenyl)methyl]-1,4-diazepane
methyl 2-[butyl(methyl)sulfamoyl]-6-(pyrazine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate