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(1R,2R)-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2,3-dihydro-1H-inden-2-ol
1-methyl-3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-(pyridin-3-ylmethyl)urea
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylurea
N-(2-fluorophenyl)-2-{4-[2-(2-methylphenoxy)acetyl]morpholin-3-yl}acetamide
dimethyl[(5-{4-[2-(pyridin-4-yl)ethyl]piperazine-1-carbonyl}-1,3,4-oxadiazol-2-yl)methyl]amine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-fluoro-4-methylphenyl)pyrrolidine-1-carboxamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-[2-(4-methoxyphenyl)phenyl]urea
3-(1-methanesulfonylpiperidin-4-yl)-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one
(2S)-1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxamide
N-methyl-1-(4-methylphenyl)-N-[(1-phenylpyrrolidin-3-yl)methyl]cyclopropane-1-carboxamide
N,N-dimethyl-3-(4-phenylbenzoyl)piperidine-1-sulfonamide
6-{2-[2-(8-fluoroquinolin-2-yl)-1H-imidazol-1-yl]ethyl}-2-methylpyrimidin-4-ol
5-chloro-2-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}phenol
5-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
N-phenyl-5-(quinoxalin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-{[(furan-2-ylmethyl)(methyl)amino]methyl}-1-[2-(piperidin-1-yl)ethyl]-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[3-(1,3-benzothiazol-2-yl)propyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-ethyl-2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
3-(2-methylphenyl)-3-phenyl-N-[2-(pyrazin-2-yl)ethyl]propanamide
8-fluoro-2-({[1-(2-hydroxyphenyl)ethyl]amino}methyl)quinolin-4-ol
N-propyl-5-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidin-2-amine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-(propan-2-yl)pyrimidine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-methylpropan-2-amine
3-(2-methoxyethyl)-1-(2-phenylethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({[(1r,4r)-4-(hydroxymethyl)cyclohexyl]methyl}sulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(3aR,5R,6S,7aS)-2-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
methyl 4-{2-amino-3-cyano-5H-chromeno[4,3-b]pyridin-4-yl}-1H-pyrazole-3-carboxylate
4-[(2-methylphenyl)methyl]-1-(2,6,8-trimethylquinoline-4-carbonyl)-1,4-diazepan-5-one
2,7,8-trimethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}quinoline-4-carboxamide
N-{3-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]phenyl}acetamide
1-(3-methoxyphenyl)-6-methyl-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-one
1-[3-(4-fluorophenoxy)propyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N3-methyl-N5-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-(1,1-dioxo-1λ6-thiolan-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-(2-ethoxyethyl)-5-[1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
[(2,4-dimethoxy-3-methylphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
(3S,9aR)-3-(2-methylpropyl)-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3R,4S)-4-(5-methylfuran-2-yl)-1-(morpholine-4-sulfonyl)pyrrolidin-3-amine
9-[(2,4-dichlorophenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(2,3-difluorophenyl)methyl]-2-{[5-(methoxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
6-(morpholin-4-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
1-(cyclopropylmethyl)-N-methyl-5-(2-methylbenzoyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-benzyl-1-(2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-3-ethyl-1,4-diazepan-5-one
N-{[1-(3-methylbutyl)pyrrolidin-3-yl]methyl}pyridine-4-carboxamide
2-phenyl-N-[1-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide