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4,5-dimethyl-2-{1-[2-(thiophen-3-yl)-1H-imidazol-1-yl]propyl}-1,3-thiazole
3-[3-(2-methoxyethyl)-5-[(2-oxoazepan-1-yl)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
(1R,3S)-3-(2-aminoethoxy)-7-(2,3-dichlorobenzoyl)-7-azaspiro[3.5]nonan-1-ol
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carboxamide
1-(2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
(2S,3R)-2-amino-1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-hydroxybutan-1-one
4-hydroxy-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(1R)-1-phenylethyl]urea
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5-methanesulfonyl-2-methylpyrimidin-4-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(quinoline-4-carbonyl)piperidin-3-ol
1-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]azepan-2-one
N-[(3S,4R)-1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(3aS,6aS)-2-methanesulfonyl-5-(3-methylbut-2-enoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 1-methoxy-2-oxo-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
(2E)-3-(3,4-dimethoxyphenyl)-N-[1-(2-phenylethyl)piperidin-3-yl]prop-2-enamide
6-methyl-2-oxo-N-[2-(pyridin-3-yloxy)propyl]-1,2-dihydropyridine-3-carboxamide
3-[(3R,4S)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
methyl 2-hydroxy-5-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]benzoate
3-fluoro-4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}morpholine
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-4-(1H-pyrazol-4-yl)butanamide
3-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(3-phenoxypropyl)pyrrolidin-3-yl]acetamide
ethyl 2-[1-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-2-yl]acetate
methyl 3-(cyclobutylmethoxy)-5-(4-methylpiperazine-1-carbonyl)benzoate
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
(4S)-3-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
6-(2,5-dimethylphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-(2-methoxypyridine-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
2-(2-chlorophenyl)-2-hydroxy-1-{7-methyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}ethan-1-one
N2-cyclopropyl-N4-methyl-N4-[2-(1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-[(4aR,7aS)-4-(2-cyclopentylacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-({5-[(3-chloro-4-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N,N-dimethyl-3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}aniline
(4aR,7aS)-N-(2-methyl-1,3-benzothiazol-5-yl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(2R)-2-amino-N,4-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pentanamide
3-{1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]piperidin-3-yl}benzoic acid
4-{[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]methyl}benzonitrile
{4-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}methanol
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
(3S,7S,8aS)-3-(hydroxymethyl)-7-({[3-(methylsulfanyl)phenyl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-(1-methylpiperidin-3-yl)-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-N-(oxan-4-yl)pyrimidin-2-amine
(4aS,7aR)-1-(2-phenylethyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,5R)-5-(pyrrolidine-1-carbonyl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
N-(3-aminopropyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methoxybenzamide