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5-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
2-(4-methoxypyrimidin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-amino-4-(1H-imidazol-4-yl)-6-methyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
1-[3-(5-benzyl-4-phenyl-1H-imidazol-1-yl)propyl]piperidin-4-ol
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-(3-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
1-(cyclohexyloxy)-3-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)propan-2-ol
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
3-{[(hexahydro-1H-pyrrolizin-7a-ylmethyl)amino]methyl}-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(methylamino)acetamide
2-[4-(5-{[(2-chlorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]propanamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(1H-pyrrol-1-yl)butanamide
5-cyclopropanecarbonyl-1'-[(2,3,5-trifluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(furan-2-ylmethyl)-2-(2-phenylethyl)-N-(prop-2-yn-1-yl)-1,3-benzoxazole-5-carboxamide
2-(3-hydroxypropyl)-9-(1-methyl-1H-pyrrole-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-methylphenyl)amino]-2-phenyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(2-hydroxy-3-methoxybenzoyl)pyrrolidine-2-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(propan-2-ylsulfanyl)phenyl]pyrrolidine-1-carboxamide
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-{4-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
(2S)-2-(methoxymethyl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
N-[(2,6-difluorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-[({1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}oxy)methyl]pyridine
2-{4-[(4-ethyl-3-oxopiperazin-1-yl)methyl]-2,6-dimethoxyphenoxy}propanoic acid
1-{2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-3-yl)propan-2-ol
1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
1-ethyl-N-[(3-methoxyphenyl)methyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-methyl-1-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-5-phenylpiperidin-2-one
3-amino-1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
(3aR,6aR)-N-{3-[(4-chlorophenyl)sulfanyl]propyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-(cyclopropylmethyl)-4-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1H-pyrazole-3-carbonyl]-2-(propan-2-yl)-1,4-diazepane
2-(2-{[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenoxy)ethan-1-ol
(1S,5R)-6-benzyl-3-[2-(4-methoxyphenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonane
({5-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-[(4-fluorophenyl)methyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
(1-{1-[(2E)-hex-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
5-methoxy-N-[1-(methoxymethyl)cyclopentyl]-3-methyl-1H-indole-2-carboxamide
4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)carbamoyl}amino)-N-(2-methoxyethyl)benzamide
1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
5-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
1-benzyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yl)propyl]acetamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide