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N-(furan-2-ylmethyl)-N-methyl-2-(thiophene-2-sulfonamido)acetamide
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
9-(2-methoxyethyl)-1-methyl-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(8-methylquinolin-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
8-(3-cyclopentylpropyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-N-(2-methoxyethyl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[(2-aminopyrimidin-5-yl)methyl]-3-chloro-4-fluoro-N-methyl-1-benzothiophene-2-carboxamide
2-(2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-4-(pyrimidin-5-yl)phenoxy)acetic acid
methyl 3-[(2-fluorophenyl)methyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2R,3R)-3-(dimethylamino)-1'-(1-ethyl-1H-pyrazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
9-[(2R)-2-hydroxy-2-(naphthalen-2-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]acetamide
2-[1-benzyl-4-(oxan-4-yl)piperazin-2-yl]ethan-1-ol
(1S,5R)-6-(cyclopropylmethyl)-3-[(4-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
4-chloro-N-{[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}aniline
4-({4-[3-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
N-{[1-(propan-2-yl)piperidin-4-yl]methyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2,5-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}furan-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(4-fluorophenoxymethyl)-1-(2-methylfuran-3-carbonyl)piperidine
2-methoxy-1-[3-(4-phenoxybenzoyl)piperidin-1-yl]ethan-1-one
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1-ethyl-1H-1,2,4-triazole
1-[(4-methylphenyl)methyl]-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazin-2-one
4-benzyl-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-3-ethyl-1,4-diazepan-5-one
2-(dimethyl-1,3-thiazol-5-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}acetamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(3-phenoxypropanoyl)pyrrolidin-3-yl]acetamide
(1S,5R)-6-benzyl-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-methyl-N-[2-(methylsulfanyl)ethyl]-3-[(pyrimidin-4-ylmethyl)sulfamoyl]benzamide
3-(3-fluorophenyl)-4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(thiophen-2-yl)propanamide
8-cyclopropanecarbonyl-2-[(4-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[2-(2,6-difluorophenyl)ethyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
N-[3-(3-methylphenyl)phenyl]-1-(pent-4-enoyl)piperidine-3-carboxamide
1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)-3-(pyridin-3-yl)propan-1-one
(5S,9aS,9bS)-5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-[3-(propan-2-yloxy)propyl]piperidin-4-amine
2-(1-methyl-1H-pyrrol-3-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
3-(2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-indole
1-(5-methoxyfuran-2-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
(4S,4aS,8aS)-4-phenyl-1-[2-(pyridin-2-yl)ethyl]-decahydroquinolin-4-ol
2-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}-3,5,7-trimethyl-1H-indole
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenyl-N-(thiophen-3-ylmethyl)benzamide
N-[1-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
2-methyl-7-[2-(1H-pyrazol-1-yl)benzoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-2-(thiophen-2-ylmethyl)propan-1-ol
N-[3-(3-chlorophenyl)phenyl]-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-4-carboxamide