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2-{1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[4-(3-hydroxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinolin-8-ol
2-(3-benzyl-1H-1,2,4-triazol-5-yl)benzonitrile
2,4-dimethyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-1,3-thiazole-5-carboxamide
N,1,3-trimethyl-N-[(3-methyloxetan-3-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
N3-[(3-fluorophenyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(2-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}(methyl)(quinoxalin-2-ylmethyl)amine
2-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidin-2-yl)pyridine
7-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2,7-diazaspiro[4.5]decane
2-(4-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperazin-1-yl)phenol
2-[(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
9-[(5-fluoro-2-methylphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2,5-dimethyl-6-[3-(2-methylphenoxy)azetidine-1-carbonyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-6-(propan-2-yl)pyridazin-3-amine
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-amine
1-[1'-(3-hydroxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
4-[1-(1H-1,2,3-benzotriazol-5-yl)-1H-imidazol-2-yl]-2-[(dimethylamino)methyl]phenol
4-ethyl-5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,3-thiazol-2-amine
2-[5-(1-ethyl-1H-indol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethan-1-ol
{[2-(5-fluoro-2-methoxyphenyl)phenyl]methyl}(propan-2-yl)amine
1,3-dimethyl-N-{[6-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-5-carboxamide
2-(1H-imidazol-1-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[2-(azepan-1-yl)ethyl]-N-ethylacetamide
1-[(5-methylfuran-2-yl)methyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-1-cyclopentylpiperidine-4-carboxamide
2-(2-oxoimidazolidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]acetamide
4-methyl-14-[4-(trifluoromethyl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-benzyl-N-(cyclobutylmethyl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
N-cyclopropyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
5-{[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
ethyl 2-{4-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]morpholin-3-yl}acetate
N-(1-methyl-1H-indazol-5-yl)-2-(pyrrolidin-3-yl)benzamide
N-methyl-2-(2-oxopiperidin-1-yl)-N-[(4-phenylphenyl)methyl]acetamide
5-(3-ethoxy-5-fluorophenyl)-6-methylpyridin-2-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylthian-4-amine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
(1S,9R)-11-[2-(2-aminoethyl)quinazolin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
3-(4-chlorophenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-phenylpropanamide
2-[({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(2-hydroxyethyl)amino]ethan-1-ol
1-cyclopentyl-N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
3-[5-({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}carbamoyl)pyridin-2-yl]benzoic acid
methyl 3-[({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)carbamoyl]benzoate